SCHEMBL7088422

SCHEMBL7088422

Cc1cc2cc(C#N)ccc2n1-c1ccc(NC(=O)c2cccnc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
POLB P06746 1/20 0.51
BRAF P15056 1/20 0.49
RAB9A P51151 7/20 0.48
CYP11B1 P15538 1/20 0.48
CYP11B2 P19099 1/20 0.48
SMN1; SMN2 Q16637 7/20 0.47
NPC1 O15118 6/20 0.47
TP53 P04637 3/20 0.47
MAPT P10636 3/20 0.47
GFER P55789 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
GAA P10253 1/20 0.47
F2 P00734 1/20 0.46
PLG P00747 1/20 0.46
PLAU P00749 1/20 0.46
KLKB1 P03952 1/20 0.46
PRSS1 P07477 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6988611 0.85 RAB9A (0.58) ALDH1A1MEN1KMT2ARAB9ASMN1; SMN2
SCHEMBL7092338 0.84 EPHX2 (0.53) ALDH1A1MEN1KMT2APOLBRAB9A
SCHEMBL6989433 0.83 ROCK2 (0.52) ALDH1A1MEN1KMT2APOLBRAB9A
SCHEMBL7139981 0.83 MEN1 (0.56) ALDH1A1MEN1KMT2APOLBBRAF
SCHEMBL7710313 0.80 HDAC1 (0.54) ALDH1A1MEN1KMT2APOLBRAB9A
SCHEMBL7707549 0.80 RAB9A (0.47) ALDH1A1MEN1KMT2APOLBRAB9A
SCHEMBL7167309 0.79 TSHR (0.49) ALDH1A1MEN1KMT2APOLBRAB9A
SCHEMBL22983039 0.79 CYP11B1 (0.74) ALDH1A1MEN1KMT2APOLBRAB9A
SCHEMBL7707527 0.78 ALDH1A1 (0.50) ALDH1A1MEN1KMT2APOLBRAB9A
SCHEMBL7707535 0.77 HDAC1 (0.50) ALDH1A1MEN1KMT2APOLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303508-A1 SUBSTITUTED 1-(4-AMINOPHENYL)INDOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2003-04-23 EP claimed
US-6353007-B1 ANTIINFLAMMATORY AGENTS AND INHIBITORS OF CELLULAR POLIFERATION BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2002-03-05 US claimed
WO-2002006273-A1 SUBSTITUTED 1-(4-AMINOPHENYL)INDOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-01-24 WO claimed
US-6353007-B1 ANTIINFLAMMATORY AGENTS AND INHIBITORS OF CELLULAR POLIFERATION BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2002-03-05 US disclosed