SCHEMBL7089033

SCHEMBL7089033

FC(F)(F)c1cc(Nc2ccc3c(c2)OCCO3)cc(C(F)(F)F)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 3/20 0.54
MAPT P10636 5/20 0.51
CNR2 P34972 1/20 0.50
ADRA2A P08913 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47
ADRA1D P25100 1/20 0.47
ADRA1A P35348 1/20 0.47
ADRA1B P35368 1/20 0.47
ULK1 O75385 1/20 0.45
KDM1A O60341 1/20 0.44
KIF11 P52732 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
AKR1C3 P42330 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24477417 0.85 TRPV1 (0.46) TRPV1MAPTCNR2KDM1AKIF11
SCHEMBL24477512 0.85 TRPV1 (0.46) TRPV1MAPTCNR2KDM1AKIF11
SCHEMBL24777901 0.82 ADRA2A (0.61) MAPTADRA2AADRA2BADRA2CADRA1D
SCHEMBL3996428 0.78 TRPV1 (0.60) TRPV1MAPTADRA2AADRA2BADRA2C
SCHEMBL4846626 0.76 TRPV1 (0.71) TRPV1MAPTADRA2AADRA2BADRA2C
SCHEMBL1009963 0.75 TRPV1 (0.62) TRPV1MAPTSMN1; SMN2MEN1KMT2A
SCHEMBL656873 0.74 SYK (0.66) ULK1
SCHEMBL394467 0.74 RAPGEF4 (0.59) MAPTKIF11AKR1C3AKR1C2
SCHEMBL657416 0.74 KDM1A (0.62) MAPTADRA2AADRA2BADRA2CADRA1D
SCHEMBL5229376 0.74 MAPT (0.81) MAPTSMN1; SMN2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1363897-A2 ANTAGONISTS OF MCP-1 FUNCTION AND METHODS OF USE THEREOF TELIK, INC. (US) 2003-11-26 EP claimed
WO-2002070509-A2 ANTAGONISTS OF MCP-1 FUNCTION AND METHODS OF USE THEREOF TELIK, INC. (US) 2002-09-12 WO claimed