SCHEMBL7089232

SCHEMBL7089232

Cc1ccccc1Nc1n[nH]c(Sc2ccc(Cl)s2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.42
LRRK2 Q5S007 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
HTT P42858 2/20 0.41
LMNA P02545 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
POLB P06746 2/20 0.41
TP53 P04637 1/20 0.41
METAP2 P50579 4/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
CCNA2 P20248 3/20 0.36
CDK2 P24941 3/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
CCNK O75909 1/20 0.36
CCND3 P30281 1/20 0.36
CDK9 P50750 1/20 0.36
CDK6 Q00534 1/20 0.36
MAPK10 P53779 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7083292 0.88 SMN1; SMN2 (0.43) PKMLRRK2SMN1; SMN2HTTLMNA
SCHEMBL7080965 0.85 SMN1; SMN2 (0.41) PKMLRRK2SMN1; SMN2HTTLMNA
SCHEMBL7090424 0.85 ALDH1A1 (0.49) PKMLRRK2SMN1; SMN2LMNANPSR1
SCHEMBL7087916 0.85 CCR4 (0.39) METAP2CCNA2CDK2CCNKCCND3
SCHEMBL5376795 0.81 METAP2 (0.41) PKMLRRK2SMN1; SMN2HTTLMNA
SCHEMBL7084630 0.80 MEN1 (0.42) SMN1; SMN2LMNAMETAP2NPC1RAB9A
SCHEMBL7088195 0.79 NFKB1 (0.48) HTTPOLBNPC1RAB9ACCNA2
SCHEMBL7085330 0.79 LRRK2 (0.43) LRRK2SMN1; SMN2HTTLMNANPSR1
SCHEMBL7089876 0.77 SMN1; SMN2 (0.44) PKMLRRK2SMN1; SMN2HTTLMNA
SCHEMBL6985036 0.75 PDE4B (0.43) SMN1; SMN2LMNANPC1RAB9ACDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1223932-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2003-01-15 EP claimed
EP-1223932-A1 COMPOUNDS AND METHODS SmithKline Beecham Corporation (US) 2002-07-24 EP claimed
WO-2001024796-A1 1,2,4-TRIAZOLE DERIVATIVES, COMPOSITION, PROCESS OF MAKING AND METHODS OF USE SMITHKLINE BEECHAM CORPORATION (US) 2001-04-12 WO claimed