SCHEMBL7089280

SCHEMBL7089280

COc1ccc(S(=O)(=O)N(Cc2ccccc2)[C@H](C(=O)OC(C)(C)C)C(C)C)cc1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 12/20 0.59
MMP9 P14780 12/20 0.59
MMP8 P22894 11/20 0.59
TAS2R14 Q9NYV8 3/20 0.56
MMP13 P45452 10/20 0.55
KEAP1 Q14145 2/20 0.54
NFE2L2 Q16236 1/20 0.54
PTGES O14684 1/20 0.54
TAS2R8 Q9NYW2 1/20 0.54
CXCR3 P49682 1/20 0.54
BMP1 P13497 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7089279 1.00 MMP2 (0.59) MMP2MMP9MMP8TAS2R14MMP13
SCHEMBL5451163 0.91 TAS2R14 (0.64) MMP2MMP9MMP8TAS2R14MMP13
SCHEMBL5097892 0.88 MMP9 (0.62) MMP2MMP9MMP8MMP13CXCR3
SCHEMBL7340794 0.88 MMP9 (0.62) MMP2MMP9MMP8MMP13CXCR3
SCHEMBL11956143 0.88 BMP1 (0.54) MMP2MMP9MMP8TAS2R14MMP13
SCHEMBL5463131 0.88 BMP1 (0.54) MMP2MMP9MMP8TAS2R14MMP13
SCHEMBL7091051 0.87 MMP2 (0.76) MMP2MMP9MMP8TAS2R14MMP13
SCHEMBL7091056 0.87 MMP2 (0.76) MMP2MMP9MMP8TAS2R14MMP13
SCHEMBL7091054 0.87 MMP2 (0.76) MMP2MMP9MMP8TAS2R14MMP13
SCHEMBL7345045 0.85 TAS2R14 (0.54) MMP2MMP9MMP8TAS2R14MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891328-B1 PEPTIDYL COMPOUNDS HAVING MMP AND TNF INHIBITORY ACTIVITY DARWIN DISCOVERY LTD (GB) 2003-08-13 EP disclosed
US-6114372-A MATRIX METALLOPROTEINASE (MMP); TUMOR NECROSIS FACTOR(TNF); COMPOUNDS SUCH AS N2-((2S)-ACETYLMERCAPTO)ACETYL-5-PHTHALIMIDOPENTANOYL)-N1-((4 -METHOXYBENZENE)SULPHONYL)-N1-(PHENYLMETHYL)HYDRAZINE DARWIN DISCOVERY LIMITED (GB) 2000-09-05 US disclosed