SCHEMBL7091327

SCHEMBL7091327

O=C(c1ccncc1)C1C2C=CC(C2)C1C(=O)c1ccncc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
HTT P42858 1/20 0.46
NAPRT Q6XQN6 1/20 0.43
GAA P10253 5/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.41
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CHRNB2 P17787 2/20 0.39
CHRNB4 P30926 2/20 0.39
CHRNA3 P32297 2/20 0.39
CHRNA4 P43681 2/20 0.39
KDM4E B2RXH2 3/20 0.39
CYP3A4 P08684 2/20 0.38
CYP2C19 P33261 2/20 0.38
MPO P05164 1/20 0.38
CYP1A2 P05177 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994870 0.80 TDP1 (0.54) POLBTDP1HTTGAAALDH1A1
SCHEMBL2140141 0.77 HTT (0.43) POLBTDP1HTTNAPRTGAA
SCHEMBL6494263 0.71 KDM4E (0.58) POLBNAPRTGAAALDH1A1MEN1
SCHEMBL6994750 0.69 CES2 (0.50) HTTALDH1A1MEN1KMT2ACHRNB2
SCHEMBL7002889 0.68 TDP1 (0.52) POLBTDP1HTTNAPRTALDH1A1
SCHEMBL28957256 0.68 POLB (0.55) POLBNAPRTGAAALDH1A1MEN1
SCHEMBL6992713 0.67 CES2 (0.48) POLBTDP1GAAALDH1A1MEN1
SCHEMBL11638730 0.67 SRD5A2 (0.58) POLBNAPRTGAAALDH1A1KDM4E
SCHEMBL18885175 0.66 NAPRT (0.39) POLBNAPRTGAAALDH1A1MEN1
SCHEMBL2985885 0.66 CHRNB2 (0.57) POLBNAPRTGAAALDH1A1CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0921119-B1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-07-02 EP disclosed
US-6114360-A Pyrrole compounds ADIR ET COMPAGNIE (FR) 2000-09-05 US disclosed
US-6063804-A Pyrrole compounds ADIR ET COMPAGNIE (FR) 2000-05-16 US disclosed
EP-0921119-A1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-06-09 EP disclosed