SCHEMBL7091666

SCHEMBL7091666

CC1=C(N)Nc2cc(C(N)C3CCCc4ccccc43)ccc2O1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PFKFB3 Q16875 1/20 0.33
IDO1 P14902 2/20 0.32
ADRA2A P08913 1/20 0.30
ADRA1D P25100 1/20 0.30
ADRA1A P35348 1/20 0.30
ADRA1B P35368 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6989617 0.99 IDO1 (0.33) PFKFB3IDO1
SCHEMBL6991849 0.94 SIGMAR1 (0.30)
Hydrochloric Acid SCHEMBL6996287 0.93 SIGMAR1 (0.31) IDO1
SCHEMBL7001764 0.79
Hydrochloric Acid SCHEMBL6998759 0.78
SCHEMBL7091667 0.74 PRMT5 (0.51) PFKFB3
Hydrochloric Acid SCHEMBL6989619 0.73 PRMT5 (0.50) PFKFB3
SCHEMBL7091668 0.71 IDO1 (0.34) IDO1TSHR
Hydrochloric Acid SCHEMBL7001640 0.69 ALOX5 (0.31)
SCHEMBL6991856 0.69 PRMT5 (0.43) ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP claimed