SCHEMBL7092175

SCHEMBL7092175

CS(=O)(=O)c1ccc(C(NC(=O)C(F)(F)F)=C(C(=O)O)c2ccc(F)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.49
AKR1C3 P42330 3/20 0.49
AKR1C2 P52895 1/20 0.49
AKR1C1 Q04828 1/20 0.49
EPHX2 P34913 4/20 0.44
FAAH O00519 1/20 0.42
MGLL Q99685 1/20 0.42
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA4 P22748 1/20 0.40
CA9 Q16790 1/20 0.40
ESR2 Q92731 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7092171 1.00 PTGS2 (0.49) PTGS2AKR1C3AKR1C2AKR1C1EPHX2
SCHEMBL7094138 0.91 PTGS2 (0.44) PTGS2AKR1C3AKR1C2AKR1C1
SCHEMBL7093579 0.91 PTGS2 (0.44) PTGS2AKR1C3AKR1C2AKR1C1
SCHEMBL7093641 0.89 AKR1C3 (0.48) PTGS2AKR1C3AKR1C2AKR1C1FAAH
SCHEMBL7092978 0.89 AKR1C3 (0.48) PTGS2AKR1C3AKR1C2AKR1C1FAAH
SCHEMBL9775660 0.77 CES1 (0.46) CA1CA9
SCHEMBL9775662 0.77 CES1 (0.46) CA1CA9
SCHEMBL7844135 0.76 PTGS2 (0.57) PTGS2AKR1C3AKR1C2AKR1C1EPHX2
SCHEMBL8092899 0.76 PTGS2 (0.57) PTGS2AKR1C3AKR1C2AKR1C1EPHX2
Carbamic Acid SCHEMBL11786852 0.72 PTGS2 (0.57) PTGS2AKR1C3AKR1C2AKR1C1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003084935-A2 DIARYL PYRIMIDINONE DERIVATIVES USEFUL FOR THE TREATMENT OF INFLAMMATION AND IMMUNOGOLICAL DISEASES ORCHID CHEMICALS & PHARMACEUTICALS LTD (IN) 2003-10-16 WO disclosed