SCHEMBL7093641

SCHEMBL7093641

CS(=O)(=O)c1ccc(/C(NC(=O)C(F)(F)F)=C(\C(=O)O)c2ccc(Cl)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 5/20 0.48
AKR1C2 P52895 1/20 0.48
AKR1C1 Q04828 1/20 0.48
MAOB P27338 2/20 0.44
PTGS2 P35354 4/20 0.43
FAAH O00519 1/20 0.41
MGLL Q99685 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
ADORA3 P0DMS8 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA2B P29275 1/20 0.39
ADORA1 P30542 1/20 0.39
MAOA P21397 1/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA9 Q16790 1/20 0.38
F2 P00734 1/20 0.38
PRSS1 P07477 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7092978 1.00 AKR1C3 (0.48) AKR1C3AKR1C2AKR1C1MAOBPTGS2
SCHEMBL7094138 0.90 PTGS2 (0.44) AKR1C3AKR1C2AKR1C1PTGS2PTGS1
SCHEMBL7093579 0.90 PTGS2 (0.44) AKR1C3AKR1C2AKR1C1PTGS2PTGS1
SCHEMBL7092171 0.89 PTGS2 (0.49) AKR1C3AKR1C2AKR1C1PTGS2FAAH
SCHEMBL7092175 0.89 PTGS2 (0.49) AKR1C3AKR1C2AKR1C1PTGS2FAAH
SCHEMBL9775662 0.76 CES1 (0.46) CA1CA9
SCHEMBL9775660 0.76 CES1 (0.46) CA1CA9
SCHEMBL13776409 0.76 AKR1C3 (0.57) AKR1C3AKR1C2AKR1C1MAOBPTGS2
SCHEMBL7641541 0.76 AKR1C3 (0.57) AKR1C3AKR1C2AKR1C1MAOBPTGS2
SCHEMBL7641537 0.76 AKR1C3 (0.57) AKR1C3AKR1C2AKR1C1MAOBPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003084935-A2 DIARYL PYRIMIDINONE DERIVATIVES USEFUL FOR THE TREATMENT OF INFLAMMATION AND IMMUNOGOLICAL DISEASES ORCHID CHEMICALS & PHARMACEUTICALS LTD (IN) 2003-10-16 WO disclosed