SCHEMBL7093579

SCHEMBL7093579

CS(=O)(=O)c1ccc(C(NC(=O)C(F)(F)F)=C(C(=O)O)c2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.44
AKR1C3 P42330 2/20 0.44
AKR1C2 P52895 1/20 0.44
AKR1C1 Q04828 1/20 0.44
PTGS1 P23219 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7094138 1.00 PTGS2 (0.44) PTGS2AKR1C3AKR1C2AKR1C1PTGS1
SCHEMBL7092175 0.91 PTGS2 (0.49) PTGS2AKR1C3AKR1C2AKR1C1
SCHEMBL7092171 0.91 PTGS2 (0.49) PTGS2AKR1C3AKR1C2AKR1C1
SCHEMBL7092978 0.90 AKR1C3 (0.48) PTGS2AKR1C3AKR1C2AKR1C1PTGS1
SCHEMBL7093641 0.90 AKR1C3 (0.48) PTGS2AKR1C3AKR1C2AKR1C1PTGS1
SCHEMBL9775662 0.87 CES1 (0.46)
SCHEMBL9775660 0.87 CES1 (0.46)
SCHEMBL5344325 0.74 PTGS2 (0.68) PTGS2AKR1C3AKR1C2AKR1C1
SCHEMBL5344331 0.74 PTGS2 (0.68) PTGS2AKR1C3AKR1C2AKR1C1
SCHEMBL5344336 0.74 PTGS2 (0.68) PTGS2AKR1C3AKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003084935-A2 DIARYL PYRIMIDINONE DERIVATIVES USEFUL FOR THE TREATMENT OF INFLAMMATION AND IMMUNOGOLICAL DISEASES ORCHID CHEMICALS & PHARMACEUTICALS LTD (IN) 2003-10-16 WO disclosed