SCHEMBL7092230

SCHEMBL7092230

COc1cccc(Cn2ccc(-c3ccco3)n2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
PKM P14618 1/20 0.49
TSHR P16473 1/20 0.49
ADORA2A P29274 4/20 0.48
ADORA1 P30542 4/20 0.48
ADORA3 P0DMS8 2/20 0.48
ADORA2B P29275 2/20 0.48
PTGS1 P23219 1/20 0.46
PTGS2 P35354 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
CD74 P04233 1/20 0.46
MIF P14174 1/20 0.46
AURKA O14965 1/20 0.45
LPO P22079 1/20 0.45
KDM4E B2RXH2 2/20 0.45
POLB P06746 1/20 0.45
RECQL P46063 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7090220 0.79 ADORA2A (0.50) ALDH1A1MEN1KMT2ATSHRADORA2A
SCHEMBL6693887 0.77 MEN1 (0.60) ALDH1A1MEN1KMT2APKMTSHR
SCHEMBL25380503 0.77 GPR55 (0.50) ALDH1A1MEN1KMT2APKMHDAC1
SCHEMBL28019857 0.76 MEN1 (0.55) ALDH1A1MEN1KMT2APKMHDAC1
SCHEMBL19086943 0.75 ALDH1A1 (0.67) ALDH1A1MEN1KMT2AHDAC1HDAC7
SCHEMBL22349826 0.72 ALDH1A1 (0.49) ALDH1A1MEN1KMT2AADORA2AADORA1
SCHEMBL28019780 0.72 MEN1 (0.50) ALDH1A1MEN1KMT2APKMHDAC1
SCHEMBL29623271 0.71 ADORA2A (0.58) ALDH1A1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL17316399 0.70 HDAC1 (0.50) ALDH1A1MEN1KMT2APKMHDAC1
SCHEMBL23923983 0.70 L3MBTL1 (0.55) MEN1KMT2APTGS2HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349552-A1 PYRAZOLO 3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055082-A1 PYRAZOLO[3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed