SCHEMBL6693887

SCHEMBL6693887

COc1cccc(Cn2cc(-c3ccco3)cn2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
ADORA2A P29274 4/20 0.53
ADORA1 P30542 4/20 0.53
ALDH1A1 P00352 5/20 0.50
PKM P14618 1/20 0.48
TSHR P16473 1/20 0.48
ADORA2B P29275 2/20 0.48
ADORA3 P0DMS8 1/20 0.48
CD74 P04233 1/20 0.47
MIF P14174 1/20 0.47
KDM4E B2RXH2 3/20 0.46
HPGD P15428 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.44
HSD17B10 Q99714 1/20 0.43
GPR55 Q9Y2T6 1/20 0.43
CMA1 P23946 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6690784 0.84 ADORA2A (0.50) ADORA2AADORA1ALDH1A1PKMADORA2B
SCHEMBL7096885 0.81 ADORA2A (0.52) MEN1KMT2AADORA2AADORA1ADORA2B
SCHEMBL7004006 0.81 L3MBTL1 (0.64) ADORA2AADORA1ALDH1A1TSHRKDM4E
SCHEMBL7096746 0.79 ADORA2A (0.54) MEN1KMT2AADORA2AADORA1ALDH1A1
SCHEMBL7092230 0.77 ALDH1A1 (0.51) MEN1KMT2AADORA2AADORA1ALDH1A1
SCHEMBL7098488 0.76 L3MBTL1 (0.57) MEN1KMT2AADORA2AADORA1ALDH1A1
SCHEMBL1703266 0.76 MEN1 (1.00) MEN1KMT2AADORA2AADORA1ALDH1A1
SCHEMBL29715635 0.76 MEN1 (1.00) MEN1KMT2AADORA2AADORA1ALDH1A1
SCHEMBL13736942 0.76 KMT2A (0.71) MEN1KMT2AADORA2AADORA1ALDH1A1
SCHEMBL4762439 0.75 MEN1 (0.69) MEN1KMT2AADORA2AADORA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2004517861-A 2004-06-17 JP claimed
EP-1349552-A1 PYRAZOLO 3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP claimed
WO-2002055082-A1 PYRAZOLO[3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO claimed