SCHEMBL7095486

SCHEMBL7095486

O=C1Nc2c[c]ccc2OC1c1ccc2c(c1)OC(F)(F)O2

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.37
NOTUM Q6P988 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CG P48736 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
MGLL Q99685 1/20 0.33
BRD4 O60885 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL910444 0.77 MMP12 (0.44)
SCHEMBL1744894 0.76 ALDH1A1 (0.39) BRD4
SCHEMBL3865428 0.72 DDB1 (0.38) RAB9ABRD4
SCHEMBL22347139 0.68 HDAC4 (0.42) HDAC4NOTUMPIK3CAPIK3CGNPC1
SCHEMBL1450577 0.68 PARP1 (0.60) BRD4
SCHEMBL20278 0.66 CTNNB1 (0.31) NOTUMPIK3CAPIK3CGNPC1RAB9A
SCHEMBL3252263 0.64 PARP1 (0.33)
SCHEMBL4267781 0.63 KDM4E (0.52) NPC1
SCHEMBL2481715 0.63 JAK1 (0.31)
SCHEMBL17634194 0.63 CA2 (0.40) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1359908-A1 QUINOLINES AND NITROGENATED DERIVATIVES THEREOF SUBSTITUTED IN 4-POSITION BY A PIPERIDINE-CONTAINING MOIETY AND THEIR USE AS ANTIBACTERIAL AGENTS SMITHKLINE BEECHAM PLC (GB) 2003-11-12 EP claimed
WO-2002056882-A1 QUINOLINES AND NITROGENATED DERIVAIVE THEREOF SUBSTITUTED IN 4-POSITION BY A PIPERIDINE-CONTAINING MOIETY AND THEIR USE AS ANTIBACTERIAL AGENTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-07-25 WO claimed