SCHEMBL7098780

SCHEMBL7098780

COc1ccccc1CCc1cnc(NC(C)c2ccccc2)nc1N

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.42
LDHA P00338 1/20 0.42
LDHB P07195 1/20 0.42
HTR7 P34969 5/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
SOS1 Q07889 2/20 0.41
DHFR P00374 1/20 0.41
EGFR P00533 1/20 0.41
KRAS P01116 1/20 0.41
ATM Q13315 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
ABCB1 P08183 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7013050 0.84 HTR7 (0.53) HTR7ADRA1DADRA1AADRA1BHDAC3
SCHEMBL7011497 0.84 ALDH1A1 (0.46) PLK1HTR7ADRA1DADRA1AADRA1B
SCHEMBL4375361 0.82 SOS1 (0.46) LDHALDHBSOS1DHFREGFR
SCHEMBL7014743 0.82 HTR7 (0.53) HTR7ADRA1DADRA1AADRA1BMEN1
SCHEMBL7010237 0.81 HTR7 (0.57) PLK1HTR7ADRA1DADRA1AADRA1B
SCHEMBL11373574 0.81 DHFR (0.58) DHFRMEN1KMT2A
SCHEMBL4374462 0.80 HTR7 (0.59) HTR7ADRA1DADRA1AADRA1B
SCHEMBL7009242 0.80 HTR7 (0.46) HTR7ADRA1DADRA1AADRA1BEGFR
SCHEMBL7011283 0.77 HTR7 (0.43) LDHALDHBHTR7ADRA1DADRA1A
SCHEMBL4375475 0.77 KMT2A (0.51) HTR7MEN1KMT2ATAAR1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1280781-A4 5-HT 7 RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2003-08-06 EP claimed
EP-1280781-A1 5-HT 7 RECEPTOR ANTAGONISTS Bristol-Myers Squibb Company (US) 2003-02-05 EP claimed
WO-2001085701-A1 5-HT7 RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-11-15 WO claimed