SCHEMBL7100181

SCHEMBL7100181

COc1ccc(Oc2ccc3c(c2)C(C(=O)O)CC(C(F)(F)F)O3)cc1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
EDNRA P25101 11/20 0.40
EDNRB P24530 10/20 0.40
PTGDR2 Q9Y5Y4 3/20 0.35
NQO2 P16083 1/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7018582 0.76 HCRTR2 (0.36) PTGS1PTGS2PTGDR2
SCHEMBL7100609 0.75 CYP11B1 (0.31) PTGS2
SCHEMBL7108605 0.74 PTGS2 (0.47) PTGS1PTGS2
SCHEMBL7019518 0.73 GRM2 (0.36) EDNRA
SCHEMBL6406090 0.70 GABRA1 (0.45) PTGS1PTGS2EDNRAEDNRBMTNR1A
SCHEMBL6413376 0.70 GABRA1 (0.45) PTGS1PTGS2EDNRAEDNRBMTNR1A
SCHEMBL7022958 0.68 GAA (0.47)
SCHEMBL6094036 0.68 PTGS2 (0.86) PTGS1PTGS2
SCHEMBL6093313 0.68 PTGS2 (0.86) PTGS1PTGS2
SCHEMBL1845395 0.66 PTGDR2 (0.49) PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1274700-A1 DIHYDROBENZOPYRANS, DIHYDROBENZOTHIOPYRANS, AND TETRAHYDROQUINOLINES FOR THE TREATMENT OF COX-2-MEDIATED DISORDERS Pharmacia Corporation (US) 2003-01-15 EP disclosed
WO-2001049675-A1 DIHYDROBENZOPYRANS, DIHYDROBENZOTHIOPYRANS, AND TETRAHYDROQUINOLINES FOR THE TREATMENT OF COX-2-MEDIATED DISORDERS PHARMACIA CORPORATION (US) 2001-07-12 WO disclosed