SCHEMBL7108605

SCHEMBL7108605

C#Cc1ccc2c(c1)C(C(=O)O)CC(C(F)(F)F)O2

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.47
PTGS1 P23219 2/20 0.47
P2RY6 Q15077 2/20 0.39
ADRA2A P08913 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30
DRD1 P21728 1/20 0.30
DRD5 P21918 1/20 0.30
OPRM1 P35372 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7018582 0.78 HCRTR2 (0.36) PTGS2PTGS1
SCHEMBL7103681 0.78 LMNA (0.35) PTGS2
SCHEMBL7019518 0.77 GRM2 (0.36)
SCHEMBL7100609 0.77 CYP11B1 (0.31) PTGS2
SCHEMBL7100181 0.74 PTGS1 (0.41) PTGS2PTGS1
SCHEMBL7167937 0.74 TSHR (0.42)
SCHEMBL7101699 0.71 ACHE (0.35) PTGS2PTGS1
SCHEMBL7171935 0.71 SMN1; SMN2 (0.47)
SCHEMBL7022958 0.69 GAA (0.47)
SCHEMBL7174724 0.69 ALDH1A1 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1274700-A1 DIHYDROBENZOPYRANS, DIHYDROBENZOTHIOPYRANS, AND TETRAHYDROQUINOLINES FOR THE TREATMENT OF COX-2-MEDIATED DISORDERS Pharmacia Corporation (US) 2003-01-15 EP disclosed
WO-2001049675-A1 DIHYDROBENZOPYRANS, DIHYDROBENZOTHIOPYRANS, AND TETRAHYDROQUINOLINES FOR THE TREATMENT OF COX-2-MEDIATED DISORDERS PHARMACIA CORPORATION (US) 2001-07-12 WO disclosed