SCHEMBL7104753

SCHEMBL7104753

N=C(N)Nc1cccc(C(=O)NC(=O)NNC(CC(=O)O)c2ccc(Cl)cc2)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 10/20 0.51
ITGAV P06756 8/20 0.51
ITGA2B P08514 6/20 0.51
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CTSA P10619 1/20 0.41
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SUCNR1 Q9BXA5 2/20 0.39
MEN1 O00255 1/20 0.39
BACE1 P56817 1/20 0.39
PARP1 P09874 1/20 0.39
PARP10 Q53GL7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7104882 0.92 ITGB3 (0.51) ITGB3ITGAVITGA2BNPC1RAB9A
SCHEMBL7099306 0.92 ITGB3 (0.51) ITGB3ITGAVITGA2BNPC1RAB9A
SCHEMBL7100982 0.90 ITGB3 (0.51) ITGB3ITGAVITGA2BNPC1RAB9A
SCHEMBL7261904 0.86 KMT2A (0.41) ITGB3ITGAVITGA2BCTSAKMT2A
SCHEMBL7105223 0.85 ITGB3 (0.55) ITGB3ITGAVITGA2BNPC1RAB9A
SCHEMBL6934969 0.81 ITGB3 (0.51) ITGB3ITGAVITGA2BNPC1RAB9A
SCHEMBL7879691 0.81 ITGB3 (0.56) ITGB3ITGAVITGA2BNPC1RAB9A
SCHEMBL7104747 0.81 CTSA (0.42) ITGB3ITGAVITGA2BNPC1RAB9A
SCHEMBL7105309 0.79 ITGB3 (0.68) ITGB3ITGAVITGA2BKMT2AMEN1
SCHEMBL13059983 0.78 ITGB3 (0.66) ITGB3ITGAVITGA2BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US claimed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP claimed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP disclosed