SCHEMBL7102639

SCHEMBL7102639

CCOC(=O)C[C@H](Cc1ccc(OCc2c(Cl)cccc2Cl)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 12/20 0.45
ITGB1 P05556 4/20 0.44
PTPN1 P18031 6/20 0.43
ATM Q13315 1/20 0.42
BCL2 P10415 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16232045 0.80 ATM (0.62) ATM
SCHEMBL4417313 0.80 ITGA4 (0.62) ITGA4ITGB1PTPN1
SCHEMBL1309887 0.80 ITGA4 (0.62) ITGA4ITGB1PTPN1
SCHEMBL838170 0.80 ITGA4 (0.62) ITGA4ITGB1PTPN1
SCHEMBL10883351 0.79 ITGA4 (0.52) ITGA4ITGB1PTPN1BCL2
SCHEMBL2779890 0.79 MMEL1 (0.62)
SCHEMBL2779899 0.79 MMEL1 (0.62)
SCHEMBL1912622 0.79 CTSS (0.55) ATMBCL2
SCHEMBL1912621 0.79 CTSS (0.55) ATMBCL2
SCHEMBL7098063 0.79 ITGA4 (0.48) ITGA4ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991619-B1 INHIBITORS OF ALPHA 4-BETA 1 MEDIATED CELL ADHESION TANABE SEIYAKU CO (JP) 2003-09-10 EP disclosed
US-6596752-B1 Small molecules that are potent inhibitors of alpha 4 beta 1 mediated adhesion to either VCAM or CS-1 and which could be useful for the treatment of inflammatory diseases. TANABE SEIYAKU CO., LTD. (JP) 2003-07-22 US disclosed
US-6482849-B1 Inhibitors of α4β1 mediated cell adhesion TANABE SEIYAKU CO., LTD. (JP) 2002-11-19 US disclosed
EP-0991619-A1 INHIBITORS OF $g(a) 4?$g(b) 1?MEDIATED CELL ADHESION TANABE SEIYAKU CO., LTD. (JP) 2000-04-12 EP disclosed
WO-1998058902-A1 INHIBITORS OF α4β1MEDIATED CELL ADHESION TANABE SEIYAKU CO., LTD. (JP) 1998-12-30 WO disclosed