SCHEMBL7102678

SCHEMBL7102678

O=CNNc1cc(Cl)cc(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 6/20 0.42
ALDH1A1 P00352 4/20 0.42
MAPT P10636 3/20 0.42
LMNA P02545 1/20 0.42
ALOX12 P18054 1/20 0.42
TSHR P16473 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
RAB9A P51151 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
FDPS P14324 1/20 0.35
DEPTOR Q8TB45 1/20 0.34
GRM4 Q14833 1/20 0.34
FADS1 O60427 1/20 0.34
FKBP1A P62942 1/20 0.33
EGFR P00533 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27675521 0.79 MAPT (0.50) GAAALDH1A1MAPTLMNAMEN1
SCHEMBL28730319 0.77 HCAR2 (0.37) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL1758240 0.76 PTGS2 (0.45) GAAALDH1A1MAPTLMNAALOX12
SCHEMBL4858206 0.76 TSHR (0.57) GAAALDH1A1MAPTLMNAALOX12
SCHEMBL2074386 0.75 ALDH1A1 (0.44) GAAALDH1A1MAPTLMNAALOX12
SCHEMBL28183482 0.71 RAPGEF4 (0.38) GAAMAPTLMNAMEN1KMT2A
SCHEMBL7151208 0.71 MEN1 (0.53) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL6755623 0.70 ALDH1A1 (0.44) ALDH1A1MAPTLMNATSHRMEN1
1,3,5-Trichlorobenzene SCHEMBL27925487 0.69 TSHR (0.47) GAAALDH1A1MAPTLMNAALOX12
SCHEMBL12838310 0.69 GAA (0.48) GAAALDH1A1MAPTLMNAALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339668-A2 BISUBSTITUTED CARBOCYCLIC CYCLOPHILIN BINDING COMPOUNDS AND THEIRUS GUILFORD PHARMACEUTICALS INC. (US) 2003-09-03 EP claimed
WO-2002044126-A2 BISUBSTITUTED CARBOCYCLIC CYCLOPHILIN BINDING COMPOUNDS AND THEIRUS GUILFORD PHARMACEUTICALS INC. (US) 2002-06-06 WO claimed