SCHEMBL7100815

SCHEMBL7100815

COc1ccc(-c2cc3cnncc3[nH]2)cc1-c1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 2/20 0.42
SMN1; SMN2 Q16637 5/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
TP53 P04637 2/20 0.42
HSD17B10 Q99714 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
ALOX15 P16050 1/20 0.42
CYP2C19 P33261 1/20 0.42
CBFB Q13951 1/20 0.42
KDM4E B2RXH2 5/20 0.41
RAB9A P51151 4/20 0.41
MAPT P10636 4/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
HTT P42858 2/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7017680 0.89 RIPK1 (0.43) RIPK1SMN1; SMN2ALDH1A1HPGDTP53
SCHEMBL7101268 0.89 RIPK1 (0.43) RIPK1SMN1; SMN2ALDH1A1HPGDTP53
SCHEMBL7101502 0.82 CCNB2 (0.44) RIPK1SMN1; SMN2ALDH1A1HPGDTP53
SCHEMBL7016833 0.82 CCNB2 (0.42) RIPK1SMN1; SMN2ALDH1A1HPGDTP53
SCHEMBL7014990 0.82 RIPK1 (0.48) RIPK1SMN1; SMN2ALDH1A1HPGDTP53
SCHEMBL5945897 0.78 ERN1 (0.49) SMN1; SMN2ALDH1A1TP53HSD17B10CYP2D6
SCHEMBL7009747 0.78 CCNB2 (0.63) RIPK1CCNB2CDK1CCNB1CCNB3
SCHEMBL7096737 0.75 NPY5R (0.45) RIPK1SMN1; SMN2ALDH1A1HPGDTP53
SCHEMBL6286924 0.75 CYP1A1 (0.44) ALDH1A1CYP3A4KDM4ERAB9AMAPT
SCHEMBL31689354 0.70 SMN1; SMN2 (0.50) SMN1; SMN2ALDH1A1HPGDTP53HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294718-A2 6,5-FUSED BICYCLIC HETEROCYCLES WARNER-LAMBERT COMPANY LLC (US) 2003-03-26 EP claimed
WO-2001096336-A2 6,5-FUSED BICYCLIC HETEROCYCLES WARNER-LAMBERT COMPANY (US) 2001-12-20 WO claimed