SCHEMBL7104882

SCHEMBL7104882

N=C(N)Nc1cccc(C(=O)NC(=O)NNC(CC(=O)O)c2cc(Cl)cc(Cl)c2)c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 8/20 0.51
ITGAV P06756 6/20 0.51
ITGA2B P08514 5/20 0.43
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PARP1 P09874 1/20 0.39
PARP10 Q53GL7 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KCNK3 O14649 1/20 0.37
KCNK9 Q9NPC2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7104753 0.92 ITGB3 (0.51) ITGB3ITGAVITGA2BNPC1RAB9A
SCHEMBL7099306 0.90 ITGB3 (0.51) ITGB3ITGAVITGA2BNPC1RAB9A
SCHEMBL7100982 0.86 ITGB3 (0.51) ITGB3ITGAVITGA2BNPC1RAB9A
SCHEMBL7104880 0.82 ITGB3 (0.43) ITGB3ITGAVITGA2BNPC1RAB9A
SCHEMBL7105223 0.82 ITGB3 (0.55) ITGB3ITGAVITGA2BNPC1RAB9A
SCHEMBL244261 0.82 ITGB3 (0.50) ITGB3ITGAVITGA2B
SCHEMBL6934969 0.81 ITGB3 (0.51) ITGB3ITGAVITGA2BNPC1RAB9A
SCHEMBL7879691 0.81 ITGB3 (0.56) ITGB3ITGAVITGA2BNPC1RAB9A
SCHEMBL4336185 0.80 ITGB3 (0.47) ITGB3ITGAVITGA2BPARP1PARP10
SCHEMBL612699 0.80 ITGB3 (0.47) ITGB3ITGAVITGA2BPARP1PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US disclosed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP disclosed