SCHEMBL7105220

SCHEMBL7105220

N=C(N)Nc1ccccc1C(=O)NC(=O)NNC(CC(=O)O)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.47
ITGAV P06756 3/20 0.47
MMP12 P39900 2/20 0.44
TDP1 Q9NUW8 1/20 0.43
EPHX1 P07099 1/20 0.39
PDE2A O00408 4/20 0.37
IGF2BP2 Q9Y6M1 1/20 0.36
FPR2 P25090 1/20 0.36
F9 P00740 1/20 0.35
ITGB5 P18084 1/20 0.35
ITGB6 P18564 1/20 0.35
ITGB8 P26012 1/20 0.35
SUCNR1 Q9BXA5 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
ITGB1 P05556 1/20 0.34
ITGA4 P13612 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7099303 0.87 KDM4E (0.43) ITGB3ITGAVITGB5ITGB6
SCHEMBL7104747 0.84 CTSA (0.42) ITGB3ITGAV
SCHEMBL7100980 0.84 ITGB3 (0.42) ITGB3ITGAV
SCHEMBL7105223 0.83 ITGB3 (0.55) ITGB3ITGAVMMP12F9
SCHEMBL7104880 0.80 ITGB3 (0.43) ITGB3ITGAV
SCHEMBL7103717 0.76 ITGB3 (0.46) ITGB3ITGAV
SCHEMBL7099306 0.69 ITGB3 (0.51) ITGB3ITGAV
SCHEMBL7099318 0.69 ITGB3 (0.42) ITGB3ITGAVITGB5ITGB6
SCHEMBL7105186 0.67 ITGB3 (0.57) ITGB3ITGAV
SCHEMBL7099324 0.67 ITGB3 (0.41) ITGB3ITGAVITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US disclosed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP disclosed