SCHEMBL7103717

SCHEMBL7103717

N=C(N)Nc1ccccc1C(=O)NC(=O)NNC(CC(=O)O)c1cccc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 4/20 0.46
ITGAV P06756 3/20 0.46
KDM4E B2RXH2 6/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
POLB P06746 1/20 0.43
ALDH1A1 P00352 4/20 0.42
PPARG P37231 1/20 0.41
HPGD P15428 2/20 0.39
HTT P42858 2/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
PTGER4 P35408 2/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
GAA P10253 1/20 0.38
LMNA P02545 1/20 0.38
ITGA2B P08514 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7099303 0.85 KDM4E (0.43) ITGB3ITGAVKDM4ESMN1; SMN2ALDH1A1
SCHEMBL7100980 0.80 ITGB3 (0.42) ITGB3ITGAVKDM4EPOLBMEN1
SCHEMBL7104747 0.80 CTSA (0.42) ITGB3ITGAVKDM4ECYP2C9CYP2C19
SCHEMBL7104880 0.80 ITGB3 (0.43) ITGB3ITGAVKDM4ESMN1; SMN2ALDH1A1
SCHEMBL7099306 0.69 ITGB3 (0.51) ITGB3ITGAVALDH1A1NPC1RAB9A
SCHEMBL7345812 0.67 BACE1 (0.47) ITGB3ITGAVKDM4EALDH1A1PPARG
SCHEMBL6778201 0.67 ITGB3 (0.52) ITGB3ITGAVITGA2B
SCHEMBL9302810 0.67 NPC1 (0.49) KDM4ESMN1; SMN2POLBALDH1A1PPARG
SCHEMBL7099318 0.66 ITGB3 (0.42) ITGB3ITGAVSMN1; SMN2ITGA2BCTSA
SCHEMBL9303274 0.66 PLAU (0.62) KDM4ESMN1; SMN2POLBCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US disclosed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP disclosed