SCHEMBL7104880

SCHEMBL7104880

N=C(N)Nc1ccccc1C(=O)NC(=O)NNC(CC(=O)O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 7/20 0.43
ITGAV P06756 6/20 0.43
DHODH Q02127 1/20 0.40
CTSA P10619 2/20 0.37
KDM4E B2RXH2 5/20 0.36
ITGA2B P08514 4/20 0.36
RECQL P46063 1/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
F10 P00742 1/20 0.35
PYGL P06737 2/20 0.34
FADS1 O60427 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7104747 0.91 CTSA (0.42) ITGB3ITGAVCTSAKDM4EITGA2B
SCHEMBL7099303 0.89 KDM4E (0.43) ITGB3ITGAVCTSAKDM4EITGA2B
SCHEMBL7100980 0.84 ITGB3 (0.42) ITGB3ITGAVKDM4EITGA2BRECQL
SCHEMBL7104882 0.82 ITGB3 (0.51) ITGB3ITGAVITGA2BALDH1A1HPGD
SCHEMBL7103717 0.80 ITGB3 (0.46) ITGB3ITGAVCTSAKDM4EITGA2B
SCHEMBL7104753 0.74 ITGB3 (0.51) ITGB3ITGAVCTSAITGA2BMEN1
SCHEMBL7099306 0.73 ITGB3 (0.51) ITGB3ITGAVITGA2BMEN1KMT2A
SCHEMBL7261894 0.70 S1PR3 (0.46) ITGB3ITGAVCTSAKDM4EITGA2B
SCHEMBL7261904 0.70 KMT2A (0.41) ITGB3ITGAVCTSAITGA2BKMT2A
SCHEMBL7099324 0.69 ITGB3 (0.41) ITGB3ITGAVITGA2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US disclosed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP disclosed