SCHEMBL7108267

SCHEMBL7108267

Cc1cc(S(C)(=O)=O)ccc1-c1ccoc(=O)c1-c1cccnc1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.46
PTGS1 P23219 4/20 0.45
ACLY P53396 2/20 0.39
LOX P28300 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7154386 0.81 MAOA (0.38) ACLY
SCHEMBL5709000 0.74 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL5708943 0.69 PTGS2 (0.58) PTGS2
SCHEMBL17205245 0.67 PTGS2 (0.59) PTGS2PTGS1CA12CA1CA2
SCHEMBL8423019 0.67 PTGS2 (0.63) PTGS2PTGS1LOXCA12CA1
SCHEMBL4940447 0.67 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL7104819 0.67 PTGS2 (0.49) PTGS2PTGS1LOX
SCHEMBL15650181 0.66 PTGS2 (0.58) PTGS2PTGS1LOXCA12CA1
SCHEMBL28111372 0.66 PTGS2 (0.58) PTGS2PTGS1
SCHEMBL7257843 0.66 PTGS2 (0.56) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1299372-A1 PYRONES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA INC. (CA) 2003-04-09 EP disclosed
WO-2002002547-A1 PYRONES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA & CO. (CA) 2002-01-10 WO disclosed