SCHEMBL7108744

SCHEMBL7108744

COc1n[c]sc1-c1nccs1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMPD3 Q9NY59 1/20 0.41
PDPK1 O15530 1/20 0.38
ECE1 P42892 1/20 0.38
CYP1A1 P04798 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP1B1 Q16678 2/20 0.33
SRC P12931 1/20 0.33
ZAP70 P43403 1/20 0.33
SYK P43405 1/20 0.33
ADRB2 P07550 1/20 0.32
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA3 P34903 1/20 0.31
GABRA2 P47869 1/20 0.31
LOXL2 Q9Y4K0 1/20 0.31
CYP2A6 P11509 1/20 0.31
FBP1 P09467 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7111538 0.70 RPS6KB2 (0.41) CYP1A2ADORA2AADORA1
SCHEMBL7458748 0.69 KDM4E (0.41) CYP1A2HSP90AA1
SCHEMBL7109776 0.69 SMPD3 (0.40) SMPD3PDPK1ECE1CYP1A1CYP1A2
SCHEMBL7108445 0.69 SMPD3 (0.40) SMPD3PDPK1ECE1CYP1A1CYP1A2
SCHEMBL468157 0.68 ALDH1A1 (0.41) CYP1A2GABRA1GABRG2GABRB3GABRA3
SCHEMBL7111032 0.68 SMPD3 (0.41) SMPD3PDPK1ECE1CYP1A1CYP1A2
SCHEMBL7105966 0.68 SMPD3 (0.39) SMPD3PDPK1ECE1CYP1A1CYP1A2
SCHEMBL10727198 0.67 PDPK1 (0.41) SMPD3PDPK1ECE1ADRB2LOXL2
SCHEMBL11148541 0.67 PDPK1 (0.42) PDPK1CYP2A6ADORA2AADORA1
SCHEMBL8613860 0.66 ALDH1A1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030008901-A1 Hydroxy pipecolate hydroxamic acid derivatives MCCLURE KIM F (US) 2003-01-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030008901-A1 Hydroxy pipecolate hydroxamic acid derivatives MMP1, MMP10, MMP3 SMPD3 1542/4885PDPK1 3673/4885ECE1 661/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.