SCHEMBL7109692

SCHEMBL7109692

CON(C)C(=O)CN1CCN(Cc2cccc(C(C)=O)c2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
KMT2A Q03164 5/20 0.48
MEN1 O00255 4/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
HSD17B10 Q99714 1/20 0.48
ATM Q13315 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HTT P42858 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
HIF1A Q16665 1/20 0.46
LMNA P02545 2/20 0.45
CHRM3 P20309 1/20 0.43
NPC1 O15118 1/20 0.43
POLB P06746 1/20 0.43
DRD4 P21917 1/20 0.43
KDM4E B2RXH2 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6864373 0.86 ALDH1A1 (0.56) ALDH1A1KMT2AMEN1HTTCYP2D6
SCHEMBL6865181 0.84 KMT2A (0.44) ALDH1A1KMT2AMEN1SMN1; SMN2HSD17B10
SCHEMBL6858172 0.83 DRD4 (0.59) ALDH1A1KMT2AMEN1SMN1; SMN2HSD17B10
SCHEMBL6864374 0.81 ALDH1A1 (0.54) ALDH1A1KMT2ASMN1; SMN2NPSR1HTT
SCHEMBL6864728 0.81 FAAH (0.53) ALDH1A1KMT2AMEN1HSD17B10CHRM3
SCHEMBL6863601 0.81 ALDH1A1 (0.59) ALDH1A1KMT2AMEN1SMN1; SMN2NPSR1
SCHEMBL7113013 0.80 CYP2D6 (0.52) ALDH1A1KMT2AMEN1SMN1; SMN2HSD17B10
SCHEMBL1481516 0.78 HDAC6 (0.58) ALDH1A1KMT2AMEN1SMN1; SMN2ATM
SCHEMBL7105308 0.78 ALDH1A1 (0.55) ALDH1A1KMT2AMEN1SMN1; SMN2HSD17B10
SCHEMBL7038584 0.76 SMN1; SMN2 (0.59) ALDH1A1KMT2AMEN1SMN1; SMN2ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US claimed
US-6800444-B1 USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS/INTERMEDIATES ISIS PHARMACEUTICALS, INC. 2004-10-05 US disclosed
US-6660466-B1 Reacting reactive appendage compounds such as meta benzylic compounds or alpha-amide compounds with scaffold molecules having reactive functionalities and contacting the intermediate library with a reducing agent ISIS PHARMACEUTICALS, INC. 2003-12-09 US disclosed
US-6150129-A USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS AND AS INTERMEDIATES FOR PREPARATION OF OTHER PHARMACEUTICAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 2000-11-21 US disclosed
US-5922872-A BACTERICIDES AND DRUGS ISIS PHARMACEUTICALS, INC. (US) 1999-07-13 US disclosed
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US disclosed
US-5798360-A ANTIBACTERIAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 1998-08-25 US disclosed
US-5780241-A ALTERING ELECTROCHEMICAL PROPERTIES BY DECYCLIZATION ISIS PHARMACEUTICALS, INC. (US) 1998-07-14 US disclosed
WO-1998020349-A1 COMPLEX CHEMICAL LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-05-14 WO disclosed
US-5731438-A BACTERICIDES; DRUGS ISIS PHARMACEUTICALS, INC. (US) 1998-03-24 US disclosed