SCHEMBL7111136

SCHEMBL7111136

O=C(NC(Cc1ccccc1)C(O)C[N+](=O)[O-])OCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 2/20 0.55
TRPM8 Q7Z2W7 1/20 0.54
CTSB P07858 6/20 0.53
CTSL P07711 5/20 0.51
SPPL2A Q8TCT8 1/20 0.49
CPA1 P15085 3/20 0.48
TACR1 P25103 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7112348 0.89 CPA1 (0.47) CTRB1TRPM8CTSBCTSLCPA1
SCHEMBL7663931 0.84 CPA1 (0.55) CPA1
SCHEMBL7810113 0.83 KLK5 (0.60) CTSBCTSL
SCHEMBL2630734 0.83 KLK5 (0.60) CTSBCTSL
SCHEMBL6861203 0.83 KLK5 (0.60) CTSBCTSL
SCHEMBL3471057 0.83 KLK5 (0.60) CTSBCTSL
SCHEMBL7111203 0.83 KLK5 (0.60) CTSBCTSL
SCHEMBL7815696 0.83 KLK5 (0.60) CTSBCTSL
SCHEMBL8838391 0.83 KLK5 (0.60) CTSBCTSL
SCHEMBL6812568 0.83 TRPM8 (0.60) CTRB1TRPM8CTSBCTSLSPPL2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030040644-A1 Synthesis of nitroalcohol diastereomers PHARM-ECO LABORATORIES, INC. 2003-02-27 US disclosed
US-6462221-B1 3-SUBSTITUTED-3-AMINO-2-HYDROXYPROPANOIC ACID SALT OR 1-NITRO-3-SUBSTITUTE-3-AMINO-2-HYDROXYPROPANOL DIASTEREOMERS OBTAINED FROM SIMULATED MOVING BED SEPARATION PHARM-ECO LABORATORIES, INC. 2002-10-08 US disclosed
EP-1159253-A2 SYNTHESIS OF NITROALCOHOL DIASTEREOMERS Johnson Matthey Pharmaceutical Materials Inc (US) 2001-12-05 EP disclosed
WO-2000050378-A9 SYNTHESIS OF NITROALCOHOL DIASTEREOMERS 2001-08-23 WO disclosed
EP-0769003-B1 AMINO ACID-DERIVED DIAMINOPROPANOLS PHARMECO LAB INC (US) 2001-05-16 EP disclosed
EP-1059285-A2 Process for the preparation of 1,3-diamino-2-propanol and 1,3-diamino-2-propanone derivatives Pharm-Eco Laboratories, Inc. (US) 2000-12-13 EP disclosed
WO-2000050378-A2 SYNTHESIS OF NITROALCOHOL DIASTEREOMERS PHARM-ECO LABORATORIES, INC. (US) 2000-08-31 WO disclosed
US-6063963-A Amino acid-derived diaminopropanols PHARM-ECO LABORATORIES, INC. (US) 2000-05-16 US disclosed
US-5631405-A Method of forming amino acid-derived diaminopropanols useful as chemical intermediates for protease-inhibitors PHARM-ECO LABORATORIES, INCORPORATED (US) 1997-05-20 US disclosed
EP-0769003-A1 AMINO ACID-DERIVED DIAMINOPROPANOLS Pharmeco Laboratories, Inc. (US) 1997-04-23 EP disclosed
US-5618966-A Method forming protease inhibitor synthetic intermediates PHARM-ECO LABORATORIES, INCORPORATED (US) 1997-04-08 US disclosed
US-5599994-A Amino acid-derived diaminopropanols PHARM-ECO LABORATORIES, INC. (US) 1997-02-04 US disclosed
WO-1996001788-A2 AMINO ACID-DERIVED DIAMINOPROPANOLS PHARM-ECO LABORATORIES, INCORPORATED (US) 1996-01-25 WO disclosed
US-5475138-A Method preparing amino acid-derived diaminopropanols PHARM-ECO LABORATORIES INCORPORATED (US) 1995-12-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030040644-A1 Synthesis of nitroalcohol diastereomers ALDH7A1, ADRA1A, ADH1A CTRB1 2741/4885TRPM8 4819/4885CTSB 4535/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.