SCHEMBL7112858

SCHEMBL7112858

CC(C)(C)C(C=O)NC(=O)c1cc(C(F)(F)F)ccc1N

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 11/20 0.44
CFTR P13569 1/20 0.44
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PTGS1 P23219 2/20 0.40
ALOX5AP P20292 4/20 0.39
FEN1 P39748 4/20 0.39
P2RX1 P51575 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7107925 0.81 PDE2A (0.39) CCR2CFTRKDM4EALDH1A1HPGD
SCHEMBL13754412 0.81 CFTR (0.48) CCR2CFTRKDM4EALDH1A1HPGD
SCHEMBL13754410 0.81 NPSR1 (0.56) CCR2CFTRKDM4EALDH1A1HPGD
SCHEMBL7109974 0.78 RXFP1 (0.51) CCR2
SCHEMBL7154000 0.77 L3MBTL1 (0.42) CCR2ALDH1A1
SCHEMBL13754426 0.76 ALOX5AP (0.57) CCR2CFTRKDM4EALDH1A1HPGD
SCHEMBL30223377 0.76 CFTR (0.54) CCR2CFTRKDM4EALDH1A1HPGD
SCHEMBL2184572 0.76 CFTR (0.54) CCR2CFTRKDM4EALDH1A1HPGD
SCHEMBL7107910 0.75 NPSR1 (0.41) CCR2PTGS1
SCHEMBL7109818 0.75 RXFP1 (0.51) CCR2KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1351924-A2 DIAMINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Bristol-Myers Squibb Pharma Company (US) 2003-10-15 EP disclosed
WO-2002050019-A2 DIAMINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB PHARMA CO. (US) 2002-06-27 WO disclosed