SCHEMBL7113291

SCHEMBL7113291

COc1ccc(-c2cc(C(F)F)nn2-c2ccc(S)c(F)c2)cc1F

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.66
PTGS1 P23219 12/20 0.66
ABCB11 O95342 1/20 0.66
ALDH1A1 P00352 1/20 0.66
KDM1A O60341 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5698611 0.89 PTGS2 (0.72) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8639053 0.84 PTGS2 (0.71) PTGS2PTGS1ABCB11ALDH1A1
Hydrogen Sulfide SCHEMBL27507738 0.83 PTGS2 (0.70) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6718470 0.82 PTGS2 (0.78) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8325061 0.81 PTGS2 (0.71) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL7876584 0.81 PTGS2 (0.73) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL24645 0.80 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8286969 0.80 PTGS2 (0.71) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL29593653 0.80 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL6601340 0.79 PTGS2 (0.98) PTGS2PTGS1ABCB11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296971-A2 2-FLUOROBENZENESULFONYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION Pharmacia Corporation (US) 2003-04-02 EP disclosed
WO-2001081332-A2 2-FLUOROBENZENESULFONYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA CORPORATION (US) 2001-11-01 WO disclosed