SCHEMBL7118232

SCHEMBL7118232

CCN(CC)CCCN(Cc1cccnc1)S(=O)(=O)c1ccc(C(N)=O)c(Nc2ccc(I)cc2)c1OCC1CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 1/20 0.35
NAMPT P43490 7/20 0.34
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
USP2 O75604 2/20 0.32
RORC P51449 1/20 0.32
ALDH1A1 P00352 3/20 0.31
GAA P10253 1/20 0.31
KDM4E B2RXH2 1/20 0.31
F2 P00734 1/20 0.31
MMP1 P03956 1/20 0.31
MMP9 P14780 1/20 0.31
MMP13 P45452 1/20 0.31
ADAM17 P78536 1/20 0.31
ADRB2 P07550 1/20 0.30
LMNA P02545 1/20 0.30
CCNA2 P20248 1/20 0.30
CDK2 P24941 1/20 0.30
CCNA1 P78396 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7118932 0.90 KMT2A (0.37) CXCR3NAMPTUSP2ALDH1A1KDM4E
SCHEMBL7120943 0.85 CXCR3 (0.34) CXCR3NAMPTUSP2RORCALDH1A1
SCHEMBL7112501 0.82 BUB1 (0.32) JAK2JAK1SYK
SCHEMBL6263086 0.81 MEN1 (0.42) CXCR3NAMPTRORCALDH1A1KDM4E
SCHEMBL6262380 0.78 CXCR3 (0.41) CXCR3NAMPTUSP2RORCALDH1A1
SCHEMBL6947384 0.78 CXCR3 (0.36) CXCR3NAMPTALDH1A1ADRB2LMNA
SCHEMBL7459563 0.77 TDP1 (0.40) CXCR3NAMPTUSP2GAAF2
SCHEMBL7122977 0.76 NAMPT (0.35) CXCR3NAMPTJAK2JAK1USP2
SCHEMBL7645897 0.74 HDAC3 (0.40) CXCR3NAMPTALDH1A1LMNAKMT2A
SCHEMBL7118222 0.74 MEN1 (0.41) ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003504401-A 2003-02-04 JP claimed
EP-1202724-A2 METHOD FOR TREATING CHRONIC PAIN USING MEK INHIBITORS WARNER-LAMBERT COMPANY (US) 2002-05-08 EP claimed
WO-2001005393-A2 METHOD FOR TREATING CHRONIC PAIN USING MEK INHIBITORS WARNER-LAMBERT COMPANY (US) 2001-01-25 WO claimed