SCHEMBL7119198

SCHEMBL7119198

CCOC(=O)c1cc(=O)c2cc(F)c(F)c(F)c2n1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.47
ALDH1A1 P00352 3/20 0.47
GAA P10253 2/20 0.47
RECQL P46063 1/20 0.44
TP53 P04637 3/20 0.44
THRB P10828 2/20 0.44
MAT2A P31153 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ALOX15 P16050 1/20 0.43
KDM4E B2RXH2 3/20 0.41
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
STAT3 P40763 1/20 0.40
ALOX12 P18054 1/20 0.40
PDE4D Q08499 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760544 0.76 MEN1 (0.53) MAPTALDH1A1GAARECQLTP53
SCHEMBL23037281 0.75 TOP2A (0.47) ALDH1A1KMT2AKDM4ESTAT3
SCHEMBL7122780 0.75 ALDH1A1 (0.43) ALDH1A1TP53KMT2AALOX15KDM4E
SCHEMBL1344450 0.74 STAT3 (0.42) MAPTALDH1A1GAARECQLTP53
SCHEMBL7123595 0.74 ALDH1A1 (0.41) MAPTALDH1A1GAAKMT2AKDM4E
SCHEMBL9870208 0.74 STAT3 (0.64) MAPTALDH1A1TP53KMT2AKDM4E
SCHEMBL22760128 0.72 MEN1 (0.51) MAPTALDH1A1GAARECQLTP53
SCHEMBL22760420 0.70 MAPT (0.47) MAPTALDH1A1GAARECQLTP53
SCHEMBL29023851 0.70 KDM4E (0.42) MAPTALDH1A1TP53KDM4EHPGD
SCHEMBL8296756 0.70 ALDH1A1 (0.63) MAPTALDH1A1GAARECQLMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
US-5763450-A BACTERICIDES; TREATMENT OF INFECTIOUS DISEASES HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP disclosed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO disclosed