SCHEMBL7123595

SCHEMBL7123595

O=C(O)c1cc(=O)c2cc(F)c(O)c(F)c2n1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
TSHR P16473 1/20 0.41
GAA P10253 2/20 0.36
AKR1C2 P52895 1/20 0.35
AKR1C1 Q04828 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPK1 P28482 2/20 0.35
KDM4E B2RXH2 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
COMT P21964 1/20 0.33
GFER P55789 1/20 0.33
AKR1B1 P15121 1/20 0.33
NOTUM Q6P988 2/20 0.33
GRN P28799 1/20 0.33
SORT1 Q99523 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7119198 0.74 MAPT (0.47) ALDH1A1GAAKMT2AKDM4ESMN1; SMN2
SCHEMBL7121568 0.73 TOP2A (0.41) ALDH1A1GAAL3MBTL1KMT2AKDM4E
SCHEMBL12984605 0.71 ALDH1A1 (0.63) ALDH1A1TSHRGAANPSR1L3MBTL1
SCHEMBL9046545 0.70 NOTUM (0.44) ALDH1A1TSHRKMT2AKDM4ESMN1; SMN2
SCHEMBL9046534 0.66 NOTUM (0.41) ALDH1A1TSHRKMT2AKDM4ESMN1; SMN2
SCHEMBL9046000 0.65 KDM4E (0.43) ALDH1A1TSHRL3MBTL1KMT2AKDM4E
SCHEMBL9044266 0.64 TDP1 (0.44) ALDH1A1TSHRL3MBTL1KMT2AKDM4E
SCHEMBL8625288 0.64 KDM4E (0.36) ALDH1A1KDM4E
SCHEMBL10668244 0.63 KDM4E (0.32) ALDH1A1KDM4E
SCHEMBL10725210 0.63 ALDH1A1 (0.34) ALDH1A1GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
US-5763450-A BACTERICIDES; TREATMENT OF INFECTIOUS DISEASES HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP disclosed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO disclosed