SCHEMBL7122780

SCHEMBL7122780

CCOC(=O)c1cc(=O)c2cc(F)c(F)c(F)c2n1C1CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.43
TSHR P16473 3/20 0.43
TOP2A P11388 1/20 0.43
TOP2B Q02880 1/20 0.43
MAPK1 P28482 2/20 0.42
KMT2A Q03164 2/20 0.39
ADRB2 P07550 1/20 0.39
KDM4E B2RXH2 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
STAT3 P40763 1/20 0.39
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
OGFRL1 Q5TC84 1/20 0.38
ALOX15 P16050 1/20 0.37
HTT P42858 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE7A Q13946 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23037281 0.94 TOP2A (0.47) ALDH1A1TSHRTOP2ATOP2BMAPK1
SCHEMBL9561861 0.84 ADRB2 (0.43) ALDH1A1TOP2ATOP2BKMT2AADRB2
SCHEMBL7844447 0.84 STAT3 (0.48) ALDH1A1TOP2ATOP2BKMT2AADRB2
SCHEMBL1345175 0.79 STAT3 (0.44) ALDH1A1TSHRTOP2ATOP2BMAPK1
SCHEMBL8096676 0.77 TOP2A (0.47) ALDH1A1TOP2ATOP2BKDM4EOPRM1
SCHEMBL9564487 0.77 MEN1 (0.43) ALDH1A1TOP2ATOP2BMAPK1KMT2A
SCHEMBL7119198 0.75 MAPT (0.47) ALDH1A1KMT2AKDM4ESTAT3ALOX15
SCHEMBL7121568 0.74 TOP2A (0.41) ALDH1A1TOP2ATOP2BKMT2AKDM4E
SCHEMBL9217647 0.73 STAT3 (0.43) ALDH1A1TSHRTOP2ATOP2BKMT2A
SCHEMBL7474321 0.73 ALDH1A1 (0.47) ALDH1A1TSHRMAPK1KMT2AOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
US-5763450-A BACTERICIDES; TREATMENT OF INFECTIOUS DISEASES HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed