SCHEMBL7120022

SCHEMBL7120022

CC(C)C(C#N)(CCC(=O)O)c1ccccc1Br

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.43
EBP Q15125 2/20 0.36
SIGMAR1 Q99720 2/20 0.36
TSHR P16473 2/20 0.35
HIF1A Q16665 2/20 0.35
CYP2C9 P11712 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
FFAR1 O14842 3/20 0.34
CYP1A2 P05177 2/20 0.33
CYP2D6 P10635 2/20 0.33
ALDH1A1 P00352 3/20 0.32
ESR1 P03372 1/20 0.31
CYP3A4 P08684 1/20 0.31
ESR2 Q92731 1/20 0.31
CYP2C19 P33261 2/20 0.31
FFAR4 Q5NUL3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7128706 0.84 L3MBTL1 (0.43) L3MBTL1EBPSIGMAR1FFAR1ALDH1A1
SCHEMBL7131088 0.84 L3MBTL1 (0.43) L3MBTL1EBPSIGMAR1TSHRFFAR1
SCHEMBL7123235 0.84 L3MBTL1 (0.43) L3MBTL1EBPSIGMAR1FFAR1ALDH1A1
SCHEMBL7129611 0.84 L3MBTL1 (0.43) L3MBTL1EBPSIGMAR1HIF1ACTSS
SCHEMBL5751980 0.81 EBP (0.51) L3MBTL1EBPSIGMAR1TSHRHIF1A
SCHEMBL10634290 0.80 L3MBTL1 (0.44) L3MBTL1EBPSIGMAR1
SCHEMBL7120088 0.78 EBP (0.40) EBPSIGMAR1TSHRHIF1ACYP2C9
SCHEMBL11823339 0.78 CTSS (0.33) TSHRHIF1ACYP2C9HSD17B10CTSS
SCHEMBL7969206 0.77 L3MBTL1 (0.40) L3MBTL1EBPSIGMAR1CYP2D6CYP3A4
SCHEMBL10631481 0.76 L3MBTL1 (0.41) L3MBTL1EBPSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6667412-B1 Carboxylic acid, ester or alcohol derivatives; n,n-substi-tuted cyclic amine or phenylacetonitrile intermediates; low cost; stability, workability, final product purity EISAI CO., LTD. (JP) 2003-12-23 US claimed
EP-1167348-A1 NITRILE DERIVATIVES Eisai Co., Ltd. (JP) 2002-01-02 EP claimed
US-6667412-B1 Carboxylic acid, ester or alcohol derivatives; n,n-substi-tuted cyclic amine or phenylacetonitrile intermediates; low cost; stability, workability, final product purity EISAI CO., LTD. (JP) 2003-12-23 US disclosed
EP-1167348-A1 NITRILE DERIVATIVES Eisai Co., Ltd. (JP) 2002-01-02 EP disclosed