SCHEMBL7128706

SCHEMBL7128706

CC(C)C(C#N)(CCC(=O)O)c1ccccc1Cl

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.43
EBP Q15125 2/20 0.36
SIGMAR1 Q99720 2/20 0.36
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
ADRA1A P35348 1/20 0.35
OPRK1 P41145 1/20 0.35
KCNH2 Q12809 1/20 0.35
KIF11 P52732 1/20 0.35
FFAR1 O14842 2/20 0.34
PTGFR P43088 3/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
POLB P06746 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MME P08473 4/20 0.32
ACE P12821 4/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7123235 0.86 L3MBTL1 (0.43) L3MBTL1EBPSIGMAR1FFAR1POLB
SCHEMBL7131088 0.84 L3MBTL1 (0.43) L3MBTL1EBPSIGMAR1FFAR1SMN1; SMN2
SCHEMBL7120022 0.84 L3MBTL1 (0.43) L3MBTL1EBPSIGMAR1FFAR1ALDH1A1
SCHEMBL7129611 0.84 L3MBTL1 (0.43) L3MBTL1EBPSIGMAR1KIF11FFAR1
SCHEMBL5751980 0.81 EBP (0.51) L3MBTL1EBPSIGMAR1KCNH2KIF11
SCHEMBL10631498 0.80 L3MBTL1 (0.44) L3MBTL1EBPSIGMAR1HTR2AHTR2C
SCHEMBL21632134 0.79 HTR2A (0.38) HTR2AHTR2CADRA1AOPRK1KCNH2
SCHEMBL11097563 0.79 FFAR1 (0.38) HTR2AHTR2CADRA1AOPRK1KCNH2
SCHEMBL7128373 0.78 MIF (0.41) L3MBTL1EBPSIGMAR1FFAR1NPC1
SCHEMBL7121340 0.77 CYP3A4 (0.39) EBPSIGMAR1HTR2AHTR2CADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6667412-B1 Carboxylic acid, ester or alcohol derivatives; n,n-substi-tuted cyclic amine or phenylacetonitrile intermediates; low cost; stability, workability, final product purity EISAI CO., LTD. (JP) 2003-12-23 US claimed
EP-1167348-A1 NITRILE DERIVATIVES Eisai Co., Ltd. (JP) 2002-01-02 EP claimed
US-6667412-B1 Carboxylic acid, ester or alcohol derivatives; n,n-substi-tuted cyclic amine or phenylacetonitrile intermediates; low cost; stability, workability, final product purity EISAI CO., LTD. (JP) 2003-12-23 US disclosed
EP-1167348-A1 NITRILE DERIVATIVES Eisai Co., Ltd. (JP) 2002-01-02 EP disclosed