SCHEMBL7123296

SCHEMBL7123296

CCOC(=O)c1cn(Cc2ccncc2)c2cc(I)ccc2c1=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 1/20 0.55
ROCK2 O75116 1/20 0.48
CDK1 P06493 1/20 0.48
PRKACA P17612 1/20 0.48
CDK2 P24941 1/20 0.48
CSNK1D P48730 1/20 0.48
GSK3A P49840 1/20 0.48
CDK5 Q00535 1/20 0.48
PRKCD Q05655 1/20 0.48
ROCK1 Q13464 1/20 0.48
CDC42BPA Q5VT25 1/20 0.48
MARK2 Q7KZI7 1/20 0.48
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.45
PTPN1 P18031 1/20 0.45
KMT2A Q03164 2/20 0.44
TDP1 Q9NUW8 1/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3003393 0.92 LMNA (0.54) P2RX3ROCK2CDK1PRKACACDK2
SCHEMBL7127566 0.85 LMNA (0.56) LMNAPTPN1CNR1CNR2
SCHEMBL1431428 0.84 LMNA (0.63) P2RX3LMNAPOLBKMT2ATDP1
SCHEMBL7120371 0.82 LMNA (0.52) P2RX3ROCK2CDK1PRKACACDK2
SCHEMBL7124395 0.81 LMNA (0.51) P2RX3ROCK2CDK1PRKACACDK2
SCHEMBL7057720 0.81 THRB (0.59) P2RX3LMNAPOLBKMT2AALDH1A1
SCHEMBL7128946 0.80 LMNA (0.52) P2RX3ROCK2CDK1PRKACACDK2
SCHEMBL5962230 0.80 LMNA (0.53) P2RX3ROCK2CDK1PRKACACDK2
SCHEMBL7120330 0.79 LMNA (0.48) P2RX3LMNAPOLBKMT2ATDP1
SCHEMBL2998174 0.79 MAP2K2 (0.52) P2RX3ROCK2CDK1PRKACACDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
US-5763450-A BACTERICIDES; TREATMENT OF INFECTIOUS DISEASES HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP disclosed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO disclosed