SCHEMBL7125719

SCHEMBL7125719

O=C(Nc1ccccc1Oc1ccc(C(=O)O)c(C(=O)O)c1)c1ccc(F)c(F)c1

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PYGM P11217 12/20 0.72
PYGL P06737 12/20 0.72
HPSE Q9Y251 1/20 0.54
TDP1 Q9NUW8 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6431898 0.90 PYGM (0.70) PYGMPYGLHPSETDP1L3MBTL1
SCHEMBL7124270 0.88 PYGL (0.66) PYGMPYGL
SCHEMBL27696838 0.88 L3MBTL1 (0.57) PYGMPYGLTDP1L3MBTL1
SCHEMBL6431208 0.87 PYGL (0.80) PYGMPYGLHPSETDP1
SCHEMBL6431433 0.86 PYGL (0.76) PYGMPYGL
SCHEMBL7125502 0.86 PYGM (0.79) PYGMPYGLHPSETDP1L3MBTL1
SCHEMBL7129478 0.86 PYGL (0.72) PYGMPYGLHPSETDP1
SCHEMBL6431607 0.85 PYGL (0.68) PYGMPYGLTDP1L3MBTL1
SCHEMBL6431424 0.85 PYGL (0.74) PYGMPYGLTDP1L3MBTL1
SCHEMBL7128870 0.85 PYGL (0.70) PYGMPYGLHPSETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030186944-A1 Such as 4-(2-(3-dimethylaminobenzoylamino)phenoxy)phthalic acid for treatment/prevention of diabetes; for inhibiting liver glycogen phosphorylase; dietetics KRISTIANSEN MARIT (DK) 2003-10-02 US disclosed
US-6590118-B1 Used in treatment of and/or prevention of diabetes, especially non-insulin dependent diabetes (Type 2 diabetes) NOVO NORDISK A/S (DK) 2003-07-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030186944-A1 Such as 4-(2-(3-dimethylaminobenzoylamino)phenoxy)phthalic acid for treatment/prevention of diabetes; for inhibiting liver glycogen phosphorylase; dietetics PYGL, GYS2, PYGM PYGM 3/4885PYGL 1/4885HPSE 1031/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.