SCHEMBL7128293

SCHEMBL7128293

O=C1N=c2ccc(CBr)cc2=N1

nearest known ligand 0.31

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
CYP4F2 P78329 1/20 0.30
CYP4A11 Q02928 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4895382 0.84 TDP1 (0.35)
SCHEMBL17423913 0.71 HSP90AA1 (0.39) CES2CES1
SCHEMBL7406780 0.69 APP (0.42)
SCHEMBL1153218 0.67 ESR1 (0.39) ALDH1A1TSHRCES2
SCHEMBL1827090 0.67 MAOA (0.37) ALDH1A1
SCHEMBL382451 0.67 NPC1 (0.35) ALDH1A1TSHR
SCHEMBL7220827 0.67
SCHEMBL3228155 0.67 KDM4E (0.35) ALDH1A1CES2CES1
SCHEMBL6345650 0.67 PARP1 (0.33) CES1
Water SCHEMBL11162060 0.65 NPC1 (0.34) ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6573379-B2 Contacting 6-methyl quinoxaline with N- bromosuccinimide in the presence of a radical initiator in 1, 2-dichloroethane to form 6-bromomethyl quinoxaline AIR PRODUCTS AND CHEMICALS, INC. 2003-06-03 US disclosed
US-20030050475-A1 Method for preparing halomethyl heterocyclic compounds BURDENIUC JUAN JESUS (US) 2003-03-13 US disclosed
EP-1277742-A1 Method for preparing halomethyl heterocyclic compounds AIR PRODUCTS AND CHEMICALS, INC. (US) 2003-01-22 EP disclosed
US-6492517-B1 THE PRESENT INVENTION RELATES TO A METHOD FOR PREPARING 5- AND 6-HALOMETHYL QUINOXALINES IN PRESENCE OF A RADICAL INITIATOR IN A SOLVENT SELECTED FROM THE GROUP CONSISTING OF FLUOROBENZENE, DIFLUOROBENZENES, TRIFLUOROBENZENES, AIR PRODUCTS AND CHEMICALS, INC. 2002-12-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030050475-A1 Method for preparing halomethyl heterocyclic compounds HDHD5, HNMT, CBR3 TRPA1 2026/4885ALDH1A1 2209/4885TSHR 1833/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.