SCHEMBL7128949

SCHEMBL7128949

CN(C)C(=O)c1ccc(C(c2ccc(Cl)cc2)N2CC(=CS(=O)(=O)Cc3cc(F)cc(F)c3)C2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 5/20 0.40
OPRM1 P35372 2/20 0.40
SLC6A9 P48067 5/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
PDK1 Q15118 1/20 0.34
FFAR2 O15552 1/20 0.33
DRD2 P14416 1/20 0.33
TBXA2R P21731 1/20 0.33
SLC6A5 Q9Y345 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK4 Q16654 1/20 0.33
GPX4 P36969 2/20 0.33
KCNH2 Q12809 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4029679 0.88 GPX4 (0.35) OPRM1SLC6A9DRD2TBXA2RGPX4
SCHEMBL3297618 0.85 GPX4 (0.34) SLC6A9GPX4
SCHEMBL3299155 0.83 GPX4 (0.34) SLC6A9GPX4KCNH2ALDH1A1
SCHEMBL3298446 0.83 GPX4 (0.34) SLC6A9GPX4KCNH2ALDH1A1
SCHEMBL7650011 0.83 FFAR2 (0.34) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7653080 0.83 FFAR2 (0.34) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3295171 0.82 HSD17B10 (0.34) SLC6A9GPX4
SCHEMBL6645535 0.81 OPRD1 (0.42) OPRD1PSEN1PSEN2APH1BNCSTN
SCHEMBL7646797 0.81 CNR1 (0.39)
SCHEMBL7652230 0.78 MEN1 (0.40) FFAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112251-B1 AZETIDINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM AVENTIS PHARMA SA (FR) 2003-05-07 EP disclosed