SCHEMBL7129435

SCHEMBL7129435

O=C(NC1NCc2ccccc21)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.51
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
OPRM1 P35372 1/20 0.47
EZH2 Q15910 1/20 0.46
SMYD3 Q9H7B4 2/20 0.42
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
LMNA P02545 2/20 0.41
ALDH1A1 P00352 1/20 0.40
DHODH Q02127 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HDAC3 O15379 1/20 0.39
CA12 O43570 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5874143 0.85 OPRM1 (0.61) HTTKMT2ASMN1; SMN2OPRM1LMNA
SCHEMBL28148420 0.81 MTNR1A (0.44) SMN1; SMN2NFKB1ALDH1A1ALOX15HDAC7
SCHEMBL7688624 0.80 GAA (0.53) HTTKMT2AMEN1SMN1; SMN2LMNA
SCHEMBL5253490 0.76 HTT (0.59) HTTKMT2AMEN1DDB1CRBN
Hydrochloric Acid SCHEMBL5186439 0.75 HTT (0.58) HTTKMT2AMEN1DDB1CRBN
SCHEMBL10920889 0.74 DRD1 (0.35) KMT2AMEN1NFKB1LMNAALDH1A1
SCHEMBL14663483 0.72 ALDH1A1 (0.62) HTTKMT2AMEN1NPC1RAB9A
SCHEMBL5573918 0.71 HDAC4 (0.35) OPRM1HDAC7TSHRNPSR1
SCHEMBL28381732 0.71 PDPK1 (0.44) KMT2AMEN1ALDH1A1HSD17B10
SCHEMBL10923547 0.71 CYP2D6 (0.38) KMT2AMEN1NFKB1ALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003231635-A MEDICINAL COMPOSITION TANABE SEIYAKU CO LTD 2003-08-19 JP disclosed
JP-2002121192-A BENZOYLAMINOISOINDOLINE DERIVATIVE, METHOD OF PRODUCING THE SAME AND INTERMEDIATE THEREFOR TANABE SEIYAKU CO LTD 2002-04-23 JP disclosed
WO-2002014276-A1 BENZOYLAMINOISOINDOLINE COMPOUNDS, PROCESSES FOR THE PREPARATION OF THE SAME AND INTERMEDIATES FOR THE SYNTHESIS THEREOF TANABE SEIYAKU CO., LTD. (JP) 2002-02-21 WO disclosed