SCHEMBL7130579

SCHEMBL7130579

COC(=O)c1ccsc1-c1cccc(O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA7 P43166 2/20 0.46
CA9 Q16790 2/20 0.46
CA14 Q9ULX7 2/20 0.46
PDK2 Q15119 1/20 0.46
PDK4 Q16654 1/20 0.46
KMT2A Q03164 4/20 0.44
MEN1 O00255 2/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
KDM4E B2RXH2 3/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
POLB P06746 1/20 0.42
ATM Q13315 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5949785 0.84 ALDH1A1 (0.50) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL3321379 0.82 KDM4E (0.56) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL5445652 0.81 PTGS1 (0.49) CA12CA1CA2CA7CA9
SCHEMBL7070888 0.81 HPGDS (0.49) CA12CA1CA2CA9HSD17B1
SCHEMBL15775647 0.80 SLC6A3 (0.53) KMT2AMEN1ALDH1A1HPGDKDM4E
SCHEMBL5949858 0.79 SLC6A4 (0.54) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL17010936 0.79 PTGS1 (0.53) KMT2AMEN1KDM4ETDP1L3MBTL1
SCHEMBL16549370 0.76 KDM4E (0.47) KMT2AMEN1ALDH1A1MAPTKDM4E
SCHEMBL7130108 0.76 KDM4E (0.43) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL7075715 0.76 KDM4E (0.43) KMT2AMEN1ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003051368-A1 N-AROYL CYCLIC AMINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2003-06-26 WO disclosed