SCHEMBL7140420

SCHEMBL7140420

COC(=O)c1ccc(C(=O)NC([C@@H]2C[C@@H](S)CN2)S(=O)(=O)c2ccc3ccccc3c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 3/20 0.44
POLB P06746 1/20 0.44
KAT6A Q92794 7/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 2/20 0.37
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36
TSHR P16473 2/20 0.36
CYP2C19 P33261 2/20 0.36
PKM P14618 2/20 0.36
MME P08473 1/20 0.36
ACE P12821 1/20 0.36
ECE1 P42892 1/20 0.36
CA2 P00918 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7141030 0.91 KAT6A (0.46) KAT6ALMNASMN1; SMN2CYP1A2CYP3A4
SCHEMBL5399404 0.91 KAT6A (0.46) KAT6ALMNASMN1; SMN2CYP1A2CYP3A4
SCHEMBL7137244 0.90 KAT6A (0.42) KAT6ALMNASMN1; SMN2PKMCA2
SCHEMBL5407300 0.90 KAT6A (0.42) KAT6ALMNASMN1; SMN2PKMCA2
SCHEMBL7148694 0.85 PKM (0.37) KAT6AALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL5422442 0.85 PKM (0.37) KAT6AALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL5409515 0.78 L3MBTL1 (0.37) MAPTLMNACYP1A2CYP3A4CYP2C9
SCHEMBL7145132 0.78 L3MBTL1 (0.37) MAPTLMNACYP1A2CYP3A4CYP2C9
SCHEMBL7146277 0.78 ACACB (0.47) KAT6AKDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL5420093 0.78 ACACB (0.47) KAT6AKDM4EALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303486-A1 PYRROLIDINE DERIVATIVES AS METALLOPROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2003-04-23 EP disclosed
WO-2002008185-A1 PYRROLIDINE DERIVATIVES AS METALLOPROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2002-01-31 WO disclosed