SCHEMBL7140857

SCHEMBL7140857

CCN(CC)c1cc(C)nc2cc(-c3ccc(CC=O)cc3)ccc12

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 4/20 0.37
NOS3 P29474 3/20 0.37
NOS2 P35228 1/20 0.37
LATS1 O95835 2/20 0.36
LATS2 Q9NRM7 2/20 0.36
CRHR1 P34998 5/20 0.34
EGLN1 Q9GZT9 1/20 0.33
DGAT1 O75907 1/20 0.32
SOAT2 O75908 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27550360 0.81 LATS1 (0.39) NOS1NOS3NOS2LATS1LATS2
SCHEMBL5400443 0.80 PGR (0.44) CRHR1EGLN1
SCHEMBL27550359 0.77 PTGS2 (0.36) LATS1LATS2CRHR1EGLN1DGAT1
SCHEMBL5409128 0.76 MAP4K4 (0.41) NOS1NOS3NOS2CRHR1
SCHEMBL7146306 0.74 NCF1 (0.53) EGLN1
SCHEMBL5419165 0.73 CRHR1 (0.42) CRHR1
SCHEMBL7137892 0.73 NCF1 (0.55) EGLN1
SCHEMBL5420608 0.73 CRHR1 (0.44) LATS1LATS2CRHR1
SCHEMBL7146671 0.71 NCF1 (0.57)
SCHEMBL14359489 0.70 NPSR1 (0.48) CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1318981-A2 QUINOLINE AND QUINAZOLINE DERIVATIVES AS LIGANDS FOR THE NEUROPEPTIDE Y RECEPTOR F. HOFFMANN-LA ROCHE AG (CH) 2003-06-18 EP disclosed
WO-2002020488-A2 QUINOLINE AND QUINAZOLINE DERIVATIVES AS LIGANDS FOR THE NEUROPEPTIDE Y RECEPTOR F. HOFFMANN-LA ROCHE AG (CH) 2002-03-14 WO disclosed