SCHEMBL7141803

SCHEMBL7141803

COC(OC)c1cc(O)ccc1[N+](=O)[O-]

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
BACE1 P56817 5/20 0.42
EGFR P00533 2/20 0.41
GPR35 Q9HC97 2/20 0.40
NPSR1 Q6W5P4 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TSHR P16473 2/20 0.38
CYP3A4 P08684 1/20 0.38
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
TXNRD1 Q16881 1/20 0.37
ALOX15 P16050 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7136446 0.81 PDK1 (0.46) ALDH1A1BACE1EGFRGPR35NPSR1
SCHEMBL2928829 0.80 MAPK1 (0.53) ALDH1A1NPSR1MAPTMAPK1TDP1
SCHEMBL5197881 0.80 ALDH1A1 (0.40) ALDH1A1EGFRMAPTTDP1TSHR
SCHEMBL11287458 0.80 TDP1 (0.53) ALDH1A1MAPTMAPK1TDP1TSHR
SCHEMBL4134840 0.80 CASP6 (0.58) ALDH1A1MAPTTSHR
SCHEMBL5196392 0.80 ALDH1A1 (0.40) ALDH1A1GPR35NPSR1MAPTMAPK1
SCHEMBL9477771 0.79 BACE1 (0.44) ALDH1A1BACE1EGFRGPR35NPSR1
SCHEMBL4125942 0.78 VCAM1 (0.55) ALDH1A1NPSR1MAPT
SCHEMBL9479720 0.75 BACE1 (0.44) ALDH1A1BACE1EGFRGPR35NPSR1
SCHEMBL7383362 0.75 ALDH1A1 (0.60) ALDH1A1GPR35NPSR1MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101035771-A 2-amino-quinazoline derivatives useful as inhibitors of beta-secretase (BACE) JANSSEN PHARMACEUTICA NV (BE) 2007-09-12 CN disclosed
US-6617456-B1 Aminoalkoxy- or hydroxyalkoxy- camptothecin compound that can be bound to a polysaccharide having carboxyl groups via an amino acid or a peptide group; antitumor agents TANABE SEIYAKU CO., LTD. (JP) 2003-09-09 US disclosed
US-6512118-B1 Pharmaceutically acceptable salt thereof show excellent antitumor activities against various tumors, especially they show excellent therapeutic effects on solid tumors such as pulmonary cancer, uterine cancer, ovarian cancer, breast TANABE SEIYAKU CO., LTD. (JP) 2003-01-28 US disclosed
EP-0781781-B1 Camptothecin derivatives TANABE SEIYAKU CO (JP) 2001-10-10 EP disclosed
US-5892043-A MIXTURE WITH POLYSACCHARIDE AND PEPTIDE; ANTITUMOR AGENT TANABE SEIYAKU CO., LTD. (JP) 1999-04-06 US disclosed
EP-0757049-B1 Camptothecin derivatives TANABE SEIYAKU CO (JP) 1999-03-24 EP disclosed
US-5847231-A Selective nitration of phenol derivatives JUNSEI CHEMICAL CO., LTD. (JP) 1998-12-08 US disclosed
US-5837673-A ANTITUMOR AGENTS AND ANTICARCINOGENIC AGENTS TANABE SEIYAKU CO., LTD. (JP) 1998-11-17 US disclosed
EP-0781781-A2 Camptothecin derivatives TANABE SEIYAKU CO., LTD. (JP) 1997-07-02 EP disclosed
EP-0757049-A1 Camptothecin derivatives TANABE SEIYAKU CO., LTD. (JP) 1997-02-05 EP disclosed