SCHEMBL7143041

SCHEMBL7143041

Cc1[nH]c2ccc(N(C(N)=S)c3ccccc3C(F)(F)F)cc2c1CCN(C)Cc1ncc([N+](=O)[O-])cn1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.34
RAB9A P51151 1/20 0.34
DRD2 P14416 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
MAPT P10636 10/20 0.33
ALDH1A1 P00352 4/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 9/20 0.32
MEN1 O00255 7/20 0.32
GAA P10253 4/20 0.32
ATM Q13315 3/20 0.32
NPSR1 Q6W5P4 2/20 0.32
CDK2 P24941 1/20 0.32
LMNA P02545 2/20 0.32
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7140896 0.94 POLB (0.34) POLBRAB9ADRD2HTR2AHTR2C
SCHEMBL8551905 0.86 ALDH1A1 (0.31) ALDH1A1
SCHEMBL8547960 0.86 ALDH1A1 (0.31) ALDH1A1
SCHEMBL8548197 0.80 HTT (0.32) ALDH1A1HTTSMN1; SMN2
SCHEMBL8548284 0.79 ALDH1A1 (0.31) ALDH1A1
SCHEMBL7146368 0.69 ALDH1A1 (0.38) POLBDRD2HTR2AHTR2CMAPT
SCHEMBL8434358 0.68 MAPT (0.33) MAPTALDH1A1KMT2AMEN1
SCHEMBL8431918 0.66 MAPT (0.34) MAPTALDH1A1KMT2AMEN1LMNA
Benzoic Acid SCHEMBL7142175 0.66 MAPT (0.34) RAB9AMAPTALDH1A1MAPK1KMT2A
SCHEMBL8589137 0.62 HTR6 (0.61) POLBDRD2HTR2AHTR2CMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0768301-B1 N-(2-substituted-3-(2-aminoethyl)-1H-indol-5-yl)-amides as new 5-HT1F agonists LILLY CO ELI (US) 2003-04-02 EP disclosed
US-6126932-A INSOLUBLE POLYMER BEARING PENDANT SIDE CHAINS, SAID SIDE CHAINS EACH TERMINATING WITH THE 1-(3-(1-PYRROLIDINYL)-PROPYL)-3-ETHYLCARBODIIMIDE MOIETY. ELI LILLY AND COMPANY (US) 2000-10-03 US disclosed
EP-0994109-A2 1-(3-(1-Pyrrolidinyl)propyl)-3-ethylcarbodiimide and a solid phase coupling agent ELI LILLY AND COMPANY (US) 2000-04-19 EP disclosed
US-5998630-A A 1-(3-(1-PYRROLIDINYL)PROPY)-3-ETHYLCARBODIIMIDE ELI LILLY AND COMPANY (US) 1999-12-07 US disclosed
WO-1997013512-A1 N-[2-SUBSTITUTED-3-(2-AMINOETHYL)-1H-INDOL-5-YL]-AMIDES: NEW 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 1997-04-17 WO disclosed
EP-0768301-A1 N-(2-substituted-3-(2-aminoethyl)-1H-indol-5-yl)-amides as new 5-HT1F agonists ELI LILLY AND COMPANY (US) 1997-04-16 EP disclosed