SCHEMBL7146381

SCHEMBL7146381

CC(=O)c1cccc(S(=O)(=O)NC(=O)Nc2c(C)cccc2C(C)(C)C)c1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.52
NLRP3 Q96P20 6/20 0.46
ALDH1A1 P00352 6/20 0.45
LMNA P02545 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.43
HTT P42858 1/20 0.41
RIPK1 Q13546 1/20 0.40
CASP3 P42574 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
FBP1 P09467 2/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7618639 0.95 KMT2A (0.47) KMT2ANLRP3ALDH1A1LMNASMN1; SMN2
SCHEMBL7137666 0.82 NLRP3 (0.67) KMT2ANLRP3HTT
SCHEMBL7146088 0.76 NLRP3 (0.73) NLRP3
SCHEMBL7141185 0.73 NLRP3 (0.72) NLRP3ALDH1A1LMNAFBP1
SCHEMBL7140924 0.73 NLRP3 (0.69) NLRP3ALDH1A1LMNAFBP1
SCHEMBL14612820 0.72 ALDH1A1 (0.67) KMT2AALDH1A1LMNASMN1; SMN2HTT
SCHEMBL7616971 0.72 NLRP3 (0.66) NLRP3
SCHEMBL11461015 0.71 NLRP3 (0.57) KMT2ANLRP3ALDH1A1LMNASMN1; SMN2
SCHEMBL7144698 0.71 NLRP3 (0.61) NLRP3
SCHEMBL4598709 0.70 SMN1; SMN2 (0.63) KMT2AALDH1A1LMNASMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0964849-B1 SULFONYL UREA DERIVATIVES AND THEIR USE IN THE CONTROL OF INTERLEUKIN-1 ACTIVITY PFIZER (US) 2003-06-04 EP disclosed
EP-1270554-A1 Sulfonyl urea derivatives and their use in the control of interleukin-1 activity PFIZER INC. (US) 2003-01-02 EP disclosed
EP-1270565-A1 4-Substituted furan-2-sulfonamide and its use in the preparation of sulfonyl urea derivatives PFIZER INC. (US) 2003-01-02 EP disclosed
US-6433009-B1 TREATMENT OF AUTOIMMUNE, CARDIOVASCULAR, NERVOUS SYSTEM, GASTROINTESTINAL, RESPIRATORY SYSTEM, AND VIRAL DISORDERS; ANTIDIABETIC, ANTIARTHRITIC, ANTIINFLAMMATORY AND ANTIDEPRESSANT AGENTS PFIZER INC 2002-08-13 US disclosed
US-6166064-A Sulfonyl urea derivatives and their use in the control of interleukin-1 activity PFIZER INC (US) 2000-12-26 US disclosed
EP-0964849-A1 SULFONYL UREA DERIVATIVES AND THEIR USE IN THE CONTROL OF INTERLEUKIN-1 ACTIVITY PFIZER INC. (US) 1999-12-22 EP disclosed
WO-1998032733-A1 SULFONYL UREA DERIVATIVES AND THEIR USE IN THE CONTROL OF INTERLEUKIN-1 ACTIVITY PFIZER INC. (US) 1998-07-30 WO disclosed