SCHEMBL4598709

SCHEMBL4598709

CC(=O)c1cccc(S(=O)(=O)NC(C)(C)C)c1

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.63
LMNA P02545 3/20 0.63
KMT2A Q03164 3/20 0.63
MAPT P10636 3/20 0.63
HPGD P15428 2/20 0.63
KDM4E B2RXH2 1/20 0.63
MEN1 O00255 1/20 0.63
NPC1 O15118 1/20 0.63
RAB9A P51151 1/20 0.63
ALDH1A1 P00352 10/20 0.60
ACLY P53396 1/20 0.49
PARG Q86W56 1/20 0.49
HTT P42858 2/20 0.46
POLB P06746 1/20 0.46
CYP19A1 P11511 1/20 0.46
TDP1 Q9NUW8 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
PKM P14618 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31426436 0.87 KDM4E (0.63) SMN1; SMN2LMNAKMT2AMAPTHPGD
SCHEMBL2568223 0.87 KDM4E (0.63) SMN1; SMN2LMNAKMT2AMAPTHPGD
SCHEMBL5041352 0.86 LMNA (0.61) SMN1; SMN2LMNAKMT2AMAPTHPGD
SCHEMBL2565620 0.84 MEN1 (0.59) SMN1; SMN2LMNAKMT2AMAPTHPGD
SCHEMBL14612820 0.83 ALDH1A1 (0.67) SMN1; SMN2LMNAKMT2AMAPTHPGD
SCHEMBL30643040 0.82 LMNA (0.56) SMN1; SMN2LMNAKMT2AMAPTHPGD
SCHEMBL26618147 0.82 LMNA (0.56) SMN1; SMN2LMNAKMT2AMAPTHPGD
SCHEMBL4057326 0.81 ALDH1A1 (0.65) SMN1; SMN2LMNAKMT2AMAPTHPGD
SCHEMBL15629008 0.80 ALDH1A1 (0.63) SMN1; SMN2LMNAKMT2AMAPTHPGD
SCHEMBL3643243 0.80 ALDH1A1 (0.58) SMN1; SMN2LMNAKMT2AMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230382889-A1 COMPOUNDS FOR INHIBITING KIF18A VOLASTRA THERAPEUTICS, INC. (US) 2023-11-30 US disclosed
US-20230382889-A1 COMPOUNDS FOR INHIBITING KIF18A VOLASTRA THERAPEUTICS, INC. (US) 2023-11-30 US disclosed
WO-2023212240-A1 COMPOUNDS FOR INHIBITING KIF18A VOLASTRA THERAPEUTICS, INC. (US) 2023-11-02 WO disclosed
US-7456195-B2 Phenylglycinamide and pyridylglycinamide derivatives useful as anticoagulants BRISTOL-MYERS SQUIBB COMPANY (US) 2008-11-25 US disclosed
US-7456195-B2 Phenylglycinamide and pyridylglycinamide derivatives useful as anticoagulants BRISTOL-MYERS SQUIBB COMPANY (US) 2008-11-25 US disclosed
EP-1910298-A2 PHENYLGLYCINAMIDE AND PYRIDYLGLYCINAMIDE DERIVATIVES USEFUL AS ANTICOAGULANTS Brystol-Myers Squibb Company (US) 2008-04-16 EP disclosed
WO-2007002313-A2 PHENYLGLYCINAMIDE AND PYRIDYLGLYCINAMIDE DERIVATIVES USEFUL AS ANTICOAGULANTS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-04 WO disclosed
US-20070003539-A1 Phenylglycinamide and pyridylglycinamide derivatives useful as anticoagulants BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-04 US disclosed
US-20070003539-A1 Phenylglycinamide and pyridylglycinamide derivatives useful as anticoagulants BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230382889-A1 COMPOUNDS FOR INHIBITING KIF18A KIF18A, KIF18B, KIF2C SMN1; SMN2 651/4885LMNA 2775/4885KMT2A 706/4885
US-20070003539-A1 Phenylglycinamide and pyridylglycinamide derivatives useful as anticoagulants F12, F11, F7 SMN1; SMN2 4597/4885LMNA 292/4885KMT2A 2453/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.