SCHEMBL7148100

SCHEMBL7148100

COc1ccc(CCCn2ccc(-c3ccsc3)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.40
KDR P35968 2/20 0.40
CYP3A4 P08684 3/20 0.39
TP53 P04637 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C9 P11712 2/20 0.39
TSHR P16473 2/20 0.39
CYP2D6 P10635 1/20 0.39
NFKB1 P19838 1/20 0.39
CYP2C19 P33261 1/20 0.39
MTOR P42345 1/20 0.39
RAB9A P51151 1/20 0.39
HIF1A Q16665 1/20 0.39
CALM1 P0DP23 1/20 0.39
MAPT P10636 3/20 0.39
TDP1 Q9NUW8 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GMNN O75496 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5754866 0.82 NPC1 (0.45) KDRCYP3A4TP53CYP1A2CYP2C9
SCHEMBL4317092 0.70 CYP17A1 (0.60) KDRFLT1FLT4GPBAR1PDGFRB
SCHEMBL5759211 0.70 SIGMAR1 (0.44) SIGMAR1MEN1KMT2AALDH1A1
SCHEMBL2780033 0.69 CYP2A6 (0.55) KDRTP53RAB9AMAPK1SMN1; SMN2
SCHEMBL10508142 0.69 MEN1 (0.69) CYP3A4TP53CYP1A2CYP2C9TSHR
SCHEMBL5757769 0.68 KDM4C (0.49) KDRFLT1FLT4PDGFRBPDGFRA
SCHEMBL22744325 0.68 CYP17A1 (0.47) TDP1
SCHEMBL244070 0.65 CALM1 (0.79) SIGMAR1CALM1TDP1MAOB
SCHEMBL4254058 0.65 CALM1 (0.72) SIGMAR1CALM1TDP1MAOB
Thiophene SCHEMBL27945185 0.65 CALM1 (0.61) SIGMAR1CALM1TDP1ALDH1A1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003500357-A 2003-01-07 JP claimed
EP-1194144-A4 ANTIBACTERIAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2002-08-07 EP claimed
EP-1194144-A1 ANTIBACTERIAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2002-04-10 EP claimed
WO-2000071120-A1 ANTIBACTERIAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2000-11-30 WO claimed