SCHEMBL7148133

SCHEMBL7148133

Nc1cccc2nc(-c3nccs3)nn12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.41
ADORA1 P30542 3/20 0.41
ADORA2B P29275 1/20 0.41
HSP90AA1 P07900 1/20 0.40
PDPK1 O15530 1/20 0.38
RAB9A P51151 5/20 0.37
NPC1 O15118 4/20 0.37
LOXL2 Q9Y4K0 1/20 0.37
AHR P35869 1/20 0.37
PKM P14618 2/20 0.36
KMT2A Q03164 2/20 0.36
RECQL P46063 1/20 0.36
TGFBR1 P36897 1/20 0.34
PDE10A Q9Y233 1/20 0.34
CYP2A6 P11509 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
METAP1 P53582 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7428889 0.77 ADORA2A (0.44) ADORA2AADORA1ADORA2BHSP90AA1RAB9A
SCHEMBL7150367 0.76 ADORA2A (0.54) ADORA2AADORA1ADORA2BNPC1KMT2A
SCHEMBL6871431 0.75 ADORA2A (0.48) ADORA2AADORA1ADORA2BPDPK1KMT2A
SCHEMBL6863122 0.74 ADORA2A (0.45) ADORA2AADORA1ADORA2B
SCHEMBL7148143 0.73 ADORA2A (0.54) ADORA2AADORA1HSP90AA1KDM4EALDH1A1
SCHEMBL6871948 0.72 HDAC2 (0.46) ADORA2ARAB9ANPC1KMT2AMEN1
SCHEMBL7144401 0.71 ADORA3 (0.53) ADORA2AADORA1ADORA2BRAB9ANPC1
SCHEMBL6868013 0.71 ADORA2A (0.42) ADORA2AADORA1ADORA2BRAB9ANPC1
SCHEMBL6872077 0.71 ADORA2A (0.42) ADORA2AADORA1ADORA2BKMT2AKDM4E
SCHEMBL6863049 0.70 ADORA2A (0.45) ADORA2AKMT2AKDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US disclosed