SCHEMBL7428889

SCHEMBL7428889

Nc1cc(Br)cc2nc(-c3nccs3)nn12

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.44
ADORA1 P30542 3/20 0.37
ADORA2B P29275 1/20 0.37
NPC1 O15118 4/20 0.36
RAB9A P51151 4/20 0.36
HSP90AA1 P07900 1/20 0.35
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 3/20 0.35
MAPT P10636 3/20 0.35
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
ABL1 P00519 1/20 0.33
BCR P11274 1/20 0.33
PDE10A Q9Y233 2/20 0.32
PKM P14618 2/20 0.32
RECQL P46063 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863122 0.80 ADORA2A (0.45) ADORA2AADORA1ADORA2BHPGD
SCHEMBL7148133 0.77 ADORA2A (0.41) ADORA2AADORA1ADORA2BNPC1RAB9A
SCHEMBL6872077 0.76 ADORA2A (0.42) ADORA2AADORA1ADORA2BKDM4EALDH1A1
SCHEMBL7427221 0.76 KDM4E (0.40) ADORA2ANPC1RAB9AKDM4EALDH1A1
SCHEMBL7429024 0.75 ADORA2A (0.39) ADORA2ANPC1RAB9AKDM4EALDH1A1
SCHEMBL6871431 0.75 ADORA2A (0.48) ADORA2AADORA1ADORA2BALDH1A1KMT2A
SCHEMBL7480280 0.75 ADORA2A (0.59) ADORA2AADORA1ADORA2BNPC1RAB9A
SCHEMBL6863814 0.74 ADORA2A (0.67) ADORA2AKDM4EHPGDABL1BCR
SCHEMBL6870494 0.74 ADORA2A (0.53) ADORA2AADORA1ADORA2BHPGDABL1
SCHEMBL6870030 0.74 ADORA2A (0.66) ADORA2AKDM4EHPGDABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP disclosed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO disclosed